Selected 5-amino-1-aryl-1H-1,2,3-triazole scaffolds as promising antiproliferative agents [PDF]
The Ukrainian Biochemical Journal, 2020 Development of a new effective drugs with low side effects and definite chemical characteristics needs indentification of bioactive scaffolds for further structural optimization.
N. Pokhodylo +3 more
doaj +1 more source
Microwave-assisted generation and reactivity of aza- and diazafulvenium methides: heterocycles via pericyclic reactions [PDF]
, 2008 Azafulvenium methides and diazafulvenium methides have been generated under microwave irradiation from 2,2-dioxo-1H,3H-pyrrolo[1,2-c]thiazoles and 2,2-dioxo-1H,3H-pyrazolo[1,5-c]thiazoles, respectively.
Melo, Teresa M. V. D. Pinho e +1 more
core +1 more source
Thiazole formation through a modified Gewald reaction
Beilstein Journal of Organic Chemistry, 2015 The synthesis of thiazoles and thiophenes starting from nitriles, via a modified Gewald reaction has been studied for a number of different substrates. 1,4-Dithiane-2,5-diol was used as the aldehyde precursor to give either 2-substituted thiazoles or 2 ...
Carl J. Mallia +3 more
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Synthesis and Biological Evaluation of Bisthiazoles and Polythiazoles
Molecules, 2018 Small heterocyclic compounds containing nitrogen and sulfur atoms, such as thiazole derivatives, represent a significant class of organic azoles that exhibit promising bioactivities and have a great potential in medicinal and agricultural fields.
Mohammed A. Al-Omair +2 more
doaj +1 more source
Structure of the cyanobactin oxidase ThcOx from Cyanothece sp. PCC 7425, the first structure to be solved at Diamond Light Source beamline I23 by means of S-SAD [PDF]
, 2016 Acknowledgements We thank Diamond Light Source for providing access to beamline I23. We also thank Thomas Sorensen and his staff for access to and support on beamline I02.
Bent, Andrew F +8 more
core +1 more source
Crystal structure of 4-(benzofuran-2-yl)-2-(3-(4-fluorophenyl)-3,3a,4,5-tetrahydro-2H-benzo[g]indazol-2-yl)thiazole, C28H20FN3OS [PDF]
, 2016 C28H20FN3OS, triclinic, P1̅ (no. 2), a = 9.5719(5) Å, b = 10.7499(6) Å, c = 10.9238(5) Å, α = 95.470(4)°, β = 102.133(4)°, γ = 97.962(4)°, V = 1079.30(10) Å3, R gt(F) = 0.0482, wR ref(F 2) = 0 ...
Abdel-Wahab, Bakr F. +4 more
core +2 more sources
The thiazole and triazole derivatives as inhibitors of metal corrosion: Part II
Zaštita Materijala, 2016 The result of the literature survey about the possibility inhibition of copper corrosion in different conditions using thiazole and triazole derivatives are presented in this review.
Đenđi Vaštag, Jelena Nakomčić
doaj +1 more source
Synthesis of various fused pyrimidine rings with their pharmacological and antimicrobial evaluation [PDF]
Journal of the Serbian Chemical Society, 2014 Various fused pyrimidine such as furo[2,3-d]pyrimidine, triazolo[1,5-a]pyrimidine, tetrazolo[1,5-a]pyrimidine were synthesized from the reactions of thioxopyrimidine-6(1H)-ones with ethyl chloroacetate (under different reaction conditions ...
Mounir Salem A. +2 more
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sp3–sp3 carbon–carbon bonds formation using 2-alkylazoles and a bromoacrylate as the reaction partners [PDF]
, 2015 International ...
Bruneau, Christian +4 more
core +3 more sources
IUCrData, 2022 The title compound, C29H25N3O3S, crystallizes in the monoclinic space group P21/n. The molecule contains a central four-ring system in which all of the rings are almost coplanar.
Sreeramapura D. Archana +5 more
doaj +1 more source