Results 11 to 20 of about 7,577,140 (312)

Inhibitory Regulation of Dendritic Activity in vivo [PDF]

open access: yesFrontiers in Neural Circuits, 2012
The spatiotemporal control of neuronal excitability is fundamental to the inhibitory process. We now have a wealth of information about the active dendritic properties of cortical neurons including axonally generated sodium action potentials as well as local sodium spikelets generated in the dendrites, calcium plateau spikes, and NMDA spikes.
Lucy Maree Palmer   +3 more
openaire   +11 more sources

Fluorine-induced polarity increases inhibitory activity of BPTI towards chymotrypsin [PDF]

open access: yes, 2022
Substituting the P1 position in bovine pancreatic trypsin inhibitor (BPTI) is known to heavily influence its inhibitory activity towards serine proteases.
Bernhard, Loll   +15 more
core   +2 more sources

Thiosemicarbazones with tyrosinase inhibitory activity [PDF]

open access: yesMedChemComm, 2019
Thiosemicarbazones reveal strong anti-tyrosinase activity.
Katarzyna Hałdys, Rafał Latajka
openaire   +2 more sources

Methoxy-Substituted Tyramine Derivatives Synthesis, Computational Studies and Tyrosinase Inhibitory Kinetics

open access: yesMolecules, 2021
Targeting tyrosinase for melanogenesis disorders is an established strategy. Hydroxyl-substituted benzoic and cinnamic acid scaffolds were incorporated into new chemotypes that displayed in vitro inhibitory effects against mushroom and human tyrosinase ...
Yasir Nazir   +7 more
doaj   +1 more source

Inhibitory Receptors Signal Activation [PDF]

open access: yesImmunity, 2008
Natural killer cell inhibitory receptors block effector responses by recruiting phosphatases that dephosphorylate molecules involved in activation. However, in this issue of Immunity, Peterson and Long show that inhibitory receptors also signal tyrosine phosphorylation, an event usually indicating cellular activation.
openaire   +2 more sources

Investigation of the inhibitory activity of extracts, fractions and secondary metabolites of Silene spp. (Caryophyllaceae) and Serratula cupuliformis (Asteraceae) on the replication of SARS-CoV-2 coronavirus

open access: yesЮг России: экология, развитие, 2023
Aim. In vitro analysis of the inhibitory activity of extracts, fractions and secondary metabolites of plants of the genus Silene [Caryophylaceae] and Serratula cupuliformis [Asteraceae) on the replication of SARS-CoV-2.Material and Methods.
E. I. Kazachinskaia   +8 more
doaj   +1 more source

Inhibitory activity of Mtb20S inhibitors.

open access: yes, 2021
Inhibitory activity of Mtb20S inhibitors.
Gang Lin (824266), Hao Zhang (15339)
core   +1 more source

Functional characterization of the Plasmodium falciparum and P-berghei homologues of macrophage migration inhibitory factor [PDF]

open access: yes, 2007
Macrophage migration inhibitory factor (MIF) is a mammalian cytokine that participates in innate and adaptive immune responses. Homologues of mammalian MIF have been discovered in parasite species infecting mammalian hosts (nematodes and malaria ...
Sarah E. Reece   +19 more
core   +1 more source

Inhibitory activity of Pf20S inhibitors and antimalarial activity.

open access: yes, 2021
Inhibitory activity of Pf20S inhibitors and antimalarial activity.
Gang Lin (824266), Hao Zhang (15339)
core   +1 more source

Synthesis and Activity against Mycobacterium tuberculosis of Olivacine and Oxygenated Derivatives

open access: yesMolecules, 2018
The tetracyclic pyrido[4,3-b]carbazole olivacine and four of its oxygenated derivatives have been synthesized by a late-stage palladium-catalyzed Heck-type cyclization of the pyrrole ring as a key step.
Ulrike Schmidt   +6 more
doaj   +1 more source

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