BLOCKADE OF M4 MUSCARINIC RECEPTORS ON STRIATAL CHOLINERGIC INTERNEURONS NORMALIZES STRIATAL DOPAMINE RELEASE IN A MOUSE MODEL OF TOR1A DYSTONIA [PDF]
, 2020 Anthony M. Downs +3 more
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Activation of Metabotropic Glutamate Receptor (mGlu2) and Muscarinic Receptors (M1, M4, and M5), Alone or in Combination, and Its Impact on the Acquisition and Retention of Learning in the Morris Water Maze, NMDA Expression and cGMP Synthesis [PDF]
, 2023 Joanna M. Wierońska +3 more
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Discovery of Selective M4 Muscarinic Acetylcholine Receptor Agonists with Novel Carbamate Isosteres
, 2019 Qingyi Yang +10 more
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Measuring ligand efficacy at the mu-opioid receptor using a conformational biosensor. [PDF]
, 2018 The intrinsic efficacy of orthosteric ligands acting at G-protein-coupled receptors (GPCRs) reflects their ability to stabilize active receptor states (R*) and is a major determinant of their physiological effects.
Livingston, Kathryn E +4 more
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Activation of the mGlu1 metabotropic glutamate receptor has antipsychotic-like effects and is required for efficacy of M4 muscarinic receptor allosteric modulators [PDF]
, 2018 Samantha E. Yohn +13 more
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Monoamine Oxidase Inhibition by Major Tanshinones from Salvia miltiorrhiza and Selective Muscarinic Acetylcholine M4 Receptor Antagonism by Tanshinone I [PDF]
, 2021 Ritu Prajapati +6 more
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Development of a Selective and High Affinity Radioligand, [3H]VU6013720, for the M4 Muscarinic Receptor [PDF]
, 2023 Aidong Qi +11 more
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An SstI polymorphism for the human muscarinic acetylchoilne receptor gene, m4 (CHRM 4)
, 1989 Sevilla D. Detera‐Wadleigh +2 more
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