Results 201 to 210 of about 8,830 (256)

Discovery of Pre-Clinical Candidate <b>VU6008055</b>/<b>AF98943</b>: A Highly Selective, Orally Bioavailable, and Structurally Distinct Tricyclic M₄ Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM) with Robust In Vivo Efficacy. [PDF]

ACS Chem Neurosci
Engers JL, Bollinger SR, Gregro AR, Capstick RA, Spearing PK, Long MF, Tarr JC, Watson KJ, Chang S, Luscombe VB, Rodriguez AL, Cho HP, Qi A, Niswender CM, Bubser M, Gould RW, Robb WH, Byun N, Gore J, Jones CK, Thomsen MS, Bridges TM, Boutaud O, Conn PJ, Engers DW, Lindsley CW, Temple KJ.   +26 more
europepmc   +1 more source

Supplementary Material for: Effects of biperiden (cholinergic muscarinic m1/m4 receptor antagonist) on craving nicotine: a proof-of-concept clinical study

karger, figshare admin, G.L.R., Ciutti, A.G., Bezerra, S., Takahashi, J.R., Jardim, R., Vicente, J.C.F., Galduróz, P., Palombo   +7 more
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Voltage-Gated and Chemogenetic Modulation of Calcium Signaling in Oligodendrocyte Development and Synaptic Integration. [PDF]

J Neurochem
Cheli VT, Paez PM.
europepmc   +1 more source

The impact of muscarinic and mGlu receptors modulators on MK-801-induced impairments in NO-dependent processes both in vitro and in vivo. [PDF]

Pharmacol Rep
Burnat G, Santocki M, Kalinowski L, Wierońska JM.   +3 more
europepmc   +1 more source

Weight Gain With Advancing Age Is Controlled by the Muscarinic Acetylcholine Receptor M4 in Male Mice.

Endocrinology
Takahashi T, Takase Y, Shiraishi A, Matsubara S, Watanabe T, Kirimoto S, Yamagaki T, Osawa M.   +7 more
europepmc   +1 more source

Regulation of m4 muscarinic receptor gene expression

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Selective labeling and localization of the M4 (m4) muscarinic receptor subtype.

Molecular Pharmacology, 1994
We report here a novel strategy for the selective labeling and localization of the M4 (m4) muscarinic receptor subtype, based on the distinct kinetics of the muscarinic antagonists dexetimide and N-methylscopolamine (NMS) and on the selectivity profile of guanylpirenzepine and AF-DX 116 for the m1-m5 muscarinic receptor subtypes expressed in CHO-K1 ...
Ferrari-Dileo, G, Waelbroeck, Magali, Mash, D C, Flynn, D D   +3 more
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Visualization of muscarinic m4 mRNA and M4 receptor subtype in rabbit lung

Life Sciences, 1993
We have used in situ hybridization to study the localization of muscarinic receptor subtype mRNAs and compared this with the distribution of muscarinic receptor subtypes using receptor autoradiography in tissue sections of the rabbit lung. To localize muscarinic receptor subtype mRNAs, subtype-specific synthetic oligonucleotide probes or riboprobes ...
Mak, JCW, Haddad, EB, Buckley, NJ, Barnes, PJ   +3 more
openaire   +4 more sources