Chemistry – A European Journal, Volume 31, Issue 8, February 6, 2025.We report the discovery of a boron‐driven ortho‐arylation reaction of N‐aryl amides and ureas. This novel method enables directed borylation of a wide range of substrates, leading to the synthesis of unique compounds such as N‐doped fulminene and diagonal tetraarylbenzenediamines.
Ganesh H. Shinde +2 more
wiley +1 more source
Visible Light-assisted Deconstruction/Refunctionalization of Strained and Unstrained N-Cycloalkylanilines [PDF]
, 2022 The exploitation of ring strain as a driving force to facilitate chemical reactions is a well-appreciated principle in organic chemistry. Of the strained carbocycles frequently explored in this respect, cyclopropane ring systems have drawn considerably ...
Boateng, Elvis Duah
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Advanced Science, Volume 12, Issue 6, February 10, 2025.A universal photoredox‐catalyzed fluoroalkylation approach by utilizing new (fluoroalkyl)diaryl methanols as versatile fluoroalkylating reagents is developed. This protocol facilitates the synthesis of mono‐, di‐, tri‐, and even polyfluoroalkylation of a broad scope of alkenes.
Heng Lu +3 more
wiley +1 more source
Development of novel methodology for the synthesis of the angucycline tetrangulol, benzo[c]phenathridines and benzonaphthopyranones [PDF]
, 2017 A thesis submitted to the Faculty of Science, University of the Witwatersrand Johannesburg. In fulfilment of the requirements for the Degree of Doctor of Philosophy.
Ngwira, Kennedy John Vijuviju
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Synthesis of aromatic heterocycles by Palladium(0)-catalyzed domino reactions and cyclization of hydrazone dianions [PDF]
This dissertation focuses on the development of new and convenient synthetic approaches for important or new aromatic heterocycles, namely chromeno[3,4-b]pyrrol-4(3H)-ones, indolo[1,2-f]phenanthridines, azaindolo[1,2-f]phenanthridines, naphtho-fused ...
Ngo, Thang Ngoc (gnd: 1123239991)
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1,3-Dien-5-ynes: Versatile Building Blocks for the Synthesis of Carbo- and Heterocycles [PDF]
, 2016 1,3-Dien-5-ynes have been extensively used as starting materials for the synthesis of a wide number of different carbo- and heterocycles. The aim of this review is to give an overview of their utility in organic synthesis, highlighting the variety of ...
Aguilar, Enrique +3 more
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Syntéza kationových helikálních N-heterocyklů [PDF]
, 2022 Diploma thesis concerns synthesis of hitherto unknown cationic helical heterocyclic compounds by catalytic processes from simple building blocks. The focus was on the utilization of a catalytic C-C bond cleavage in biphenylene followed by annulation with
Hrubý, Samuel
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Mise en évidence d'une résistance aux trypanocides parmi des souches de Trypanosoma congolense récemment isolées au Burkina [PDF]
, 1984 Dix-huit souches de T. congolense ont fait l'objet d'une épreuve de sensibilité à l'acétate de diminazène et à l'isométamidium chez la souris. L'intérêt et les limites de cette épreuve sont discutés. Les 13 souches de T.
Authié, Edith
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Visible Light-Induced Green Synthesis of Phenanthridines via C—H Activation of Simple Alkanes [PDF]
, 2021 Wenyi Li, Wei‐Min He
openalex +1 more source
Trypanosoma brucei aquaglyceroporin 2 is a high-affinity transporter for pentamidine and melaminophenyl arsenic drugs and the main genetic determinant of resistance to these drugs [PDF]
, 2017 Objectives Trypanosoma brucei drug transporters include the TbAT1/P2 aminopurine transporter and the high-affinity pentamidine transporter (HAPT1), but the genetic identity of HAPT1 is unknown. We recently reported that loss of T. brucei aquaglyceroporin
Aguinaga Andrés, David +19 more
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