Results 101 to 110 of about 1,467 (158)

Carrier cross-reactivities of the bile acid reabsorption inhibitors elobixibat, linerixibat, maralixibat, and odevixibat. [PDF]

J Lipid Res
Billo V, Neelen C, Wannowius M, Neubauer A, Fühler B, Hagos Y, Geyer J.   +6 more
europepmc   +1 more source

Comment on the article: "Microvascular effects of intravenous esmolol in patients with normal cardiac function undergoing postoperative atrial fibrillation: a prospective pilot study in cardiothoracic surgery". [PDF]

Crit Care, 2019
Zheng YY, Guo F, Lu B, Li Q.
europepmc   +1 more source

Predicting compounds that interact with the 2 known agonist-induced conformations of the human β1-adrenoceptor. [PDF]

Mol Pharmacol
Baker JG, Lim VJY, Proudman RGW, Giese FNZ, Kolb P.   +4 more
europepmc   +1 more source

Early Intravenous Beta-Blockade with Esmolol in Adults with Severe Traumatic Brain Injury (EBB-TBI): Protocol for a Phase 2a Intervention Design Study. [PDF]

Neurocrit Care
Thomas M, Hayes K, White P, Ramesh A, Culliford L, Ackland G, Pickering A.   +6 more
europepmc   +1 more source

Potent drug delivery enhancement of betulinic acid and NVX-207 into equine skin in vitro - a comparison between a novel oxygen flow-assisted transdermal application device and microemulsion gels. [PDF]

BMC Vet Res
Zscherpe P, Kalbitz J, Weber LA, Paschke R, Mäder K, von Rechenberg B, Cavalleri JV, Meißner J, Klein K.   +8 more
europepmc   +1 more source

Biting behaviour, spatio-temporal dynamics, and the insecticide resistance status of malaria vectors in different ecological zones in Ghana. [PDF]

Parasit Vectors
Akuoko OK, Dhikrullahi SB, Hinne IA, Mohammed AR, Owusu-Asenso CM, Coleman S, Dadzie SK, Kyerematen R, Boakye DA, Wilson MD, Afrane YA.   +10 more
europepmc   +1 more source

Effects of carvedilol on human prostate tissue contractility and stromal cell growth pointing to potential clinical implications. [PDF]

Pharmacol Rep
Hu S, Müderrisoglu AE, Ciotkowska A, Kale O, Keller P, Schott M, Tamalunas A, Waidelich R, Stief CG, Hennenberg M.   +9 more
europepmc   +1 more source

Enzyme catalyzed stereoselective synthesis of (S)-propanolamines

Tetrahedron: Asymmetry, 1994
Abstract Stereoselective synthesis of (S)-propanolamines has been carried out by the ring opening of racemic epoxides with 2-propylamine in presence of lipases and subtilisin. The effect of solvent towards selectivity has also been studied.
Ahmed Kamal
exaly   +3 more sources

o-Chlorobenzenesulfonamidic derivatives of (aryloxy)propanolamines as .beta.-blocking/diuretic agents

Journal of Medicinal Chemistry, 1993
A series of compounds 1b-f, 2b-f, and 3b-f having an o-chlorobenzenesulfonamidic diuretic moiety variously linked to the nitrogen side chain of the beta-blocking (aryloxy)propanolamine pharmacophore were prepared and tested for their beta 1-adrenoceptor ...
Violetta Cecchetti, Arnaldo Fravolini, Oriana Tabarrini   +2 more
exaly   +5 more sources

Role of the (acyloxy)methyl moiety in eliciting the adrenergic .beta.-blocking activity of 3-(acyloxy)propanolamines

Journal of Medicinal Chemistry, 1987
Some totally aliphatic 3-(acyloxy)propanolamines were synthesized with the aim of testing whether @blocking activity could be obtained from this class of drugs, even in the absence of an aromatic group.
B Macchia, Annalina Lapucci, Adriano Martinelli   +2 more
exaly   +4 more sources