Elucidating the roles of TM7SF3 and LHFPL6 in the putative H +/OC antiporter function in the human brain capillary endothelial cell line, hCMEC/D3. [PDF]
INTRODUCTION: The putative proton/organic cation (H +/OC) antiporter has been shown to mediate transport of CNS drug compounds like oxycodone and pyrilamine across the blood-brain barrier (BBB).
Schmid, Benjamin +9 more
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Histamine H1-receptor-mediated keratan sulfate production in rabbit chondrocytes: involvement of protein kinase C [PDF]
, 1991 We investigated the characteristics of the histamine H1-receptor in cultured rabbit chondrocytes. Scatchard analysis of [3H]pyrilamine, an H1-antagonist, binding to the chondrocytes revealed a single class of binding sites with KD and Bmax values of 90 +/
T. Kuno +6 more
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Effect of histamine H1 and H2 receptor antagonists on histamine-induced macrophage LOX-1 mRNA expression. [PDF]
, 2014 Monocyte-derived macrophages were incubated in the presence of 10 µM histamine and the indicated concentrations of the histamine H1 and H2 receptor antagonists (pyrilamine and ranitidine, respectively) for 4 h and analyzed for LOX-1 mRNA expression.
Petri T. Kovanen (188189) +3 more
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Characterization of histamine receptors mediating contraction and relaxation of the ovarian follicle wall [PDF]
, 1987 Histamine is known to be present in ovarian tissue and may play a role in the ovulation process. The effect of histamine on the follicular smooth musculature was investigated using strips from the protruding part of mature bovine follicles, mounted in ...
Owman, Ch +3 more
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The role of histamine receptors on rabbit articular chondrocytes [PDF]
, 1991 Using the radioligand histamine H_1 antagonist [^3H] -pyrilamine and H_2 antagonist [^3H] -tiotidine, we characterized the histamine H_1 and H_2 receptors on rabbit articular chondrocytes.
Matsumura, Fuminori, 松村, 文典
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Vasopeptidase-activated latent ligands of the histamine receptor-1 [PDF]
, 2013 Whether peptidases present in vascular cells can activate prodrugs active on vascular cells has been tested with 2 potential latent ligands of the histamine H1 receptor (H1R). First, a peptide consisting of the antihistamine cetirizine (CTZ) condensed at
Marceau, François +3 more
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EFFECTS OF H1- AND H2- RECEPTOR ANTAGONISTS ON THE HISTAMINE- AND HISTAMINE AGONISTS- INDUCED RESPONSE IN THE ISOLATED GUINEA PIG INTESTINE DURING ONTOGENY [PDF]
, 1990 THE PURPOSE OF THE PRESENT INVESTIGATION WAS TO STUDY THE EFFECTS OF H1- AND H2- ANTAGONISTS ON THE CONTRACTIONS INDUCED BY HISTAMINE AS WELL AS BY HISTAMINE AGONISTS IN INTESTINAL SMOOTH MUSCLE OF GUINEA PIG DURING DEVELOPMENT.
Koutsoviti-Papadopoulou, Maria +1 more
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Cerrahpaşa Medical Journal, 2019 The aim of the study is to determine the effects of histamine receptors on the ileum smooth muscle contractions and the role of nitric oxide on these effects.
Aşkın HEKİMOĞLU, Ramazan ÇİÇEK
doaj
The immunological release of slow-reacting substance of anaphylaxis from bovine lung [PDF]
LR: 20061115; PUBM: Print; JID: 0372712; 0 (Prostaglandins); 0 (SRS-A); 361-37-5 (Methysergide); 50-67-9 (Serotonin); 50-78-2 (Aspirin); 51-45-6 (Histamine); 51-55-8 (Atropine); 9014-72-6 (Polyphloretin Phosphate); 91-84-9 (Pyrilamine); ppublishSource ...
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Indomethacin-antihistamine combination for gastric ulceration control [PDF]
, 1981 An anti-inflammatory and analgesic composition containing indomethacin and an H sub 1 or an H sub 2 histamine receptor antagonist in an amount sufficient to reduce gastric distress caused by the indomethacin is described.
Brown, P. A., Danellis, J. V.
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