Results 111 to 120 of about 822,055 (188)

Circulating tumour DNA in mCRPC: bridging tumour biology and real-time treatment monitoring. [PDF]

Front Mol Med
Kaoma C, Sathekge M, Chalwe J, Mokoala K, Kgatle M.   +4 more
europepmc   +1 more source

A Preliminary Evaluation of ¹⁷⁷Lu-PSMA-617-Based Targeted Radioligand Therapy with X-Ray Stimulated PSMA Relocation Using the <i>PiggyBac</i> Reporter-Gene-Engineered Orthotopic Prostate Tumor Model. [PDF]

Pharmaceutics
Chen YT, Huang KH, Wu CY, Lee YJ.
europepmc   +1 more source

Peptidomics and pharmacological profiling of Odontobuthus doriae (Buthidae) scorpion venom at the kappa opioid receptor. [PDF]

Sci Rep
Abdollahnia A, Bata BB, Fraunhofer A, Hermes J, Atashi J, Ghassempour A, Gruber CW.   +6 more
europepmc   +1 more source

A Holistic Approach to Identifying a Positron Emission Tomography (PET) Tracer Candidate for In Vivo Imaging of Purinergic P2X7 Receptor in Neuroinflammation. [PDF]

ACS Pharmacol Transl Sci
Ghafir El Idrissi I, Spinaci A, Vitone D, Intranuovo F, Niso M, Brunetti L, Francucci B, Pazarlar BA, Magnusdottir KH, Paradies E, Marobbio CMT, Ricci L, Grignolo M, Iacobazzi RM, Marucci G, Dal Ben D, Lambertucci C, Volpini R, Denora N, Adinolfi E, Mikkelsen JD, Buccioni M, Lacivita E, Leopoldo M.   +23 more
europepmc   +1 more source

Structural basis of opioid receptor activation by PCP and ketamine. [PDF]

Nat Struct Mol Biol
Jiang Q, Han J, Fine EJ, Ramos-Gonzalez N, Rangari VA, Ruiz MV, Critz ML, Suomivuori CM, Wang J, Albert TL, Whiddon K, Li K, Robertson MJ, Huang XP, Land BB, Majumdar S, Fay JF, Dror RO, Che T.   +18 more
europepmc   +1 more source

Using a NanoBRET-Based Ligand-Binding Assay at the β₂-Adrenoceptor for Undergraduate Pharmacology Education. [PDF]

Pharmacol Res Perspect
Pearce A, Huang X, Redfern-Nichols T, Sisk CM, Safitri D, Collins M, Malcharek MA, García ST, Nakamura C, Harris A, Ladds G.   +10 more
europepmc   +1 more source

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia. [PDF]

Sci Adv
Wang Y, Luo P, Xu H, Zhan L, Sakamoto K, Li M, Wang J, Huang XP, Zhou J, Liu T, Suo Y, Fan W, He X, Xu Y, Cai Y, Wang C, Zhao Y, Dai A, Lai Y, Yuan Q, Hu W, Wu K, Yang D, Cheng X, Lu X, Krumm B, Kenakin T, Zhang J, Roth BL, Gao Z, Xu HE, Zhuang Y.   +31 more
europepmc   +1 more source

Affinity-Tuned Albumin Hitchhiking Extends the Bioorthogonal Capture Window in Pretargeting Radiotheranostics. [PDF]

Adv Healthc Mater
He X, Fletcher NL, Ediriweera GR, Zhu Y, Humphries J, Howard CB, Wang J, Bell CA, Kempe K, Thurecht KJ.   +9 more
europepmc   +1 more source

A Ligand-Triggered Receptor Conformation Enables the Design of Selective Agonists for the Dopamine 3 Receptor (D₃R) Using a Bitopic Strategy. [PDF]

JACS Au
Arroyo-Urea S, Nazarova AL, Knieb A, Abdulsalam H, Jahan K, Du T, Gao S, Newman AH, Katritch V, García-Nafría J, Bonifazi A.   +10 more
europepmc   +1 more source

Emerging Insights into the Distinct Pharmacological Mechanisms of Buprenorphine. [PDF]

J Chem Inf Model
Alonso-Carrasco A, Quintana-Garcia A, Ciruela-Jardí M, Casadó-Anguera V, Enten GA, Llopart N, Carrasco-Martinez B, Cai NS, Moreno E, Ferré S, Casadó V, Pardo L.   +11 more
europepmc   +1 more source