Results 151 to 160 of about 3,259,253 (212)

Peptidomics and pharmacological profiling of Odontobuthus doriae (Buthidae) scorpion venom at the kappa opioid receptor. [PDF]

Sci Rep
Abdollahnia A, Bata BB, Fraunhofer A, Hermes J, Atashi J, Ghassempour A, Gruber CW.   +6 more
europepmc   +1 more source

A Preliminary Evaluation of ¹⁷⁷Lu-PSMA-617-Based Targeted Radioligand Therapy with X-Ray Stimulated PSMA Relocation Using the <i>PiggyBac</i> Reporter-Gene-Engineered Orthotopic Prostate Tumor Model. [PDF]

Pharmaceutics
Chen YT, Huang KH, Wu CY, Lee YJ.
europepmc   +1 more source

A Holistic Approach to Identifying a Positron Emission Tomography (PET) Tracer Candidate for In Vivo Imaging of Purinergic P2X7 Receptor in Neuroinflammation. [PDF]

ACS Pharmacol Transl Sci
Ghafir El Idrissi I, Spinaci A, Vitone D, Intranuovo F, Niso M, Brunetti L, Francucci B, Pazarlar BA, Magnusdottir KH, Paradies E, Marobbio CMT, Ricci L, Grignolo M, Iacobazzi RM, Marucci G, Dal Ben D, Lambertucci C, Volpini R, Denora N, Adinolfi E, Mikkelsen JD, Buccioni M, Lacivita E, Leopoldo M.   +23 more
europepmc   +1 more source

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia. [PDF]

Sci Adv
Wang Y, Luo P, Xu H, Zhan L, Sakamoto K, Li M, Wang J, Huang XP, Zhou J, Liu T, Suo Y, Fan W, He X, Xu Y, Cai Y, Wang C, Zhao Y, Dai A, Lai Y, Yuan Q, Hu W, Wu K, Yang D, Cheng X, Lu X, Krumm B, Kenakin T, Zhang J, Roth BL, Gao Z, Xu HE, Zhuang Y.   +31 more
europepmc   +1 more source

Structural basis of opioid receptor activation by PCP and ketamine. [PDF]

Nat Struct Mol Biol
Jiang Q, Han J, Fine EJ, Ramos-Gonzalez N, Rangari VA, Ruiz MV, Critz ML, Suomivuori CM, Wang J, Albert TL, Whiddon K, Li K, Robertson MJ, Huang XP, Land BB, Majumdar S, Fay JF, Dror RO, Che T.   +18 more
europepmc   +1 more source

Neuropharmacology of levamisole and its phase I metabolites: lack of evidence for levamisole-cocaine interactions. [PDF]

Psychopharmacology (Berl)
Zolkowska D, Lehner KR, Partilla JS, Blough BE, Baumann MH.   +4 more
europepmc   +1 more source

Using a NanoBRET-Based Ligand-Binding Assay at the β₂-Adrenoceptor for Undergraduate Pharmacology Education. [PDF]

Pharmacol Res Perspect
Pearce A, Huang X, Redfern-Nichols T, Sisk CM, Safitri D, Collins M, Malcharek MA, García ST, Nakamura C, Harris A, Ladds G.   +10 more
europepmc   +1 more source

Characterization of binding properties to human P-glycoprotein: development of a [3H]verapamil radioligand-binding assay.

Journal of Pharmacology and Experimental Therapeutics, 1999
Interaction with the exsorptive transporter P-glycoprotein (P-gp) is a possible source of peculiarities in drug pharmacokinetics, including dose-dependent absorption, drug-drug interactions, intestinal secretion, and limited permeability of the blood ...
S. Döppenschmitt, P. Langguth, C. Regårdh, T. Andersson, C. Hilgendorf, H. Spahn-Langguth   +5 more
semanticscholar   +2 more sources