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Rilpivirine in HIV-1-positive women initiating pregnancy: to switch or not to switch?
, 2020 International audienceBackgroundSafety data about rilpivirine use during pregnancy remain scarce, and rilpivirine plasma concentrations are reduced during second/third trimesters, with a potential risk of viral breakthroughs.Benoist, Laurence, Blondin, Gilles, Mohamed, Khaled, Chiarello, Pierre, Peretti, Delphine, Djoubou, Sandrine, Bailly-Salin, Philippe, Rey, David, Fayolas, Isabelle, Godinot, Matthieu, Pannier, Emmanuelle, Le Chenadec, Jérôme, Floch-Tudal, Corinne, Gerbe, Juliette, Matheron, Sophie, Hau, Isabelle, Vaucel, Edouard, Firtion, Ghislaine, Lavarenne, Gaelle, Samar, Ketty, Rivaux, Danièle, Perfezou, Pascale, Bobrie-Moyrand, Claire, Bourdic, Katia, Niault, Mathilde, Jabbarian, Hélène, David, Selva, Laine, Laeticia, Lebrette, Marie-Gisèle, Meier, Françoise, Ceccaldi, Pierre-François, Garion, Dominique, Fontelonga, Marie-Agnès, Lachassine, Eric, Lafeuillade, Alain, Clech, Laure, Tubiana, Roland, Brunet-Cartier, Cécile, Lévy, Marc, Pauchard, Michèle, Marcou, Valerie, Carré, Nathalie, Mazy, Fabienne, Schmit, Jean-Luc, Dupre, Christelle, Genet, Philippe, Partisani, Marialuisa, Chevry, Coralie, Gaillat, Jacques, Mortier, Emmanuel, Warszawski, Josiane, Schmidt, Jean-Luc, Sandler, Boris, Elharrar, Brigitte, Lalande, Muriel, Cudeville, Corinne, Barat, Muriel, Gilbert, Sylvie, Elleau, Christophe, Boissinot, Christine, Sanchez, Audrey, Johnson, Ama, Agher, Nouara, Ichou, Houria, Khuong-Josses, Marie-Aude, Calin, Ruxandra-Oana, Elbert, Véronique Lefevre, Monnier, Sylvie, Yahia, Fatma Ait, D’angelo, Sophie, Garnier-André, Elisabeth, Guigue, Nelly, Sahadatu, Osseni, Khadly, Redouane, Fleury, Hervé, Picard, Fabienne, Touboul, Claudine, Dollfus, Catherine, Ogoudjobi, Stanislas, Kayem, Gilles, Karaoui, Leïla, Hatchuel, Yves, Ronat, Véronique, Ajana, Faiza, Pluchart, Claire, Reynes, Jacques, Masse, Virginie, Jacquier, Françoise, Vanderbergh, Anne, Dukiel, Nathalie, Poinsignon, Yves, Guerin-Duplessy, Anne, Briquet, Catherine, Winter, Cécile, Devidas, Alain, Roca, Didier, Debruyne, Elise, Ducrocq, Sarah, Fernandes, Elisabeth, Malbrunot, Claire, Brouard, Jacques, Dommergues, Marc, Moreau, Laurence, Salmon-Ceron, Dominique, Runel-Belliard, Camille, Hammou, Yamina, Muanza, Blandine, Zakaria, Ahmed, Courdavault, Laurence, Bouldouyre, Marie-Anne, Moine, Agnès Bourgeois, Cheneau, Christine, Vintejoux, Emmanuelle, Benbara, Amélie, Brunel-Dalmas, Florence, Allouche, Claude, Chacé, Anne, Vaillant, Odile Luycx, Huri, Virginie, Damond, Florence, Alixe, Véronique, Matheron, Isabelle, Garrait, Valérie, Esnault, Jean-Luc, Bernard, Louis, Joras, Marine, Catteau, Odile, Chiabrando, Julie, Bouabdallah, Soufiane, Castaneda, Julie, Diallo, Mama Doufari, Ducroix-Roubertou, Sophie, Bonmarchand, Manuela, Richier, Laurent, Narcy, Catherine, Samama, Déborah, Billiemaz, Kareen, Nourry, Christelle, Galvan, Valérie, Dauphin, Hélène, Launay, Odile, Boquet, Laurence, Bajawi, Youcef, Rouzioux, Christine, Hubert, Claire, Foucaud, Pierre, Fialaire, Pascale, Frange, Pierre, Allal, Lahcene, de Morel, Philippe, Vaudre, Geneviève, Partizani, Marialuisa, Lefort, Agnès, Andris, Sabine, Ranaivojaona, Sata, Leverger, Guy, Palenzuela, Gilles, Goubin, Pascale, Guimard, Thomas, Carpentier, Bénédicte, Daniel, Corinne, Ouamara-Digue, Enora, Armand, Evelyne, Shneider, Luminata, Checoury, Alain, Brault, Dominique, Levine, Martine, Canestri, Ana, Boumediene, Marie Astride, Brossier, Jean-Pierre, Errichiello, Katia, Langer, Bruno, Cravello, Ludovic, Etienne, Lise, Durand, Myriam, Osman, Zafer, Gardiennet, Quentin, Goussef, Marie, Abbal, Julie, Labrune, Philippe, Paquiez, Odile, Cayla, Claudine, Rohan, Jennifer, Rouger, Christine, Maraux, Barbara, Pinquier, Didier, Borgne, Anne, Makhloufi, Djamila, Grelier, Anne, Bachelard, Germaine, Bertrand, Yves, Carbillon, Lionel, Decaux, Nathalie, Nemeth, Céline, Wifaq, Bouchra, Lambry, Véronique, Borie, Constance, Martha, Sandrine-Anne, Allisy, Christine, Le Coz, Marie-Françoise, Bongain, André, Colombani, Dominique, Belzic, Isabelle, Donnadieu, Anne-Claire, Duthé, Jean-Charles, Caby, Fabienne, Piet, Emilie, Rajguru, Mandovi, Nassar, Rania, Winer, Norbert, Mouton-Rioux, Virginie, Chambrin, Véronique, Zarouk, Virginie, Raho-Moussa, Mariem, Bogner, Noëlle, Beucher, Gaël, Crenn-Hebert, Catherine, Medus, Marie, Aubry, Olivier, Le Moine, Philippe, Delannoy, Catherine, Ebel, Edith, Dos-Santos, Emmanuelle, Uettwiller, Françoise, Jabbar, Ahmed, Fourcade, Corinne, Ferry, A., Louchard, Agnès, Blanc-Ruffat, Isabelle, Genet, Claire, Boiron, Emilie, Brun, Jean-Luc, Fanget, Cécile, Vitrat, Virginie, Deschaud, Martine, Zebelus, Jenny, Heller-Roussin, Brigitte, Mourey, Marie-Christine, Sanchez, Anita, Francoise, Michel, Nahri, Imad, Reliquet, Véronique, Mousset, Gaetane, Carbonnel-Delalande, Elisabeth, Avettand-Fenoël, Véronique, Dendale-Nguyen, Joëlle, Leveille, Sandrine, Schmitt, Marie Paule, Rodallec, Audrey, Nisand, Israël, Bellahcene, Chahrazede, Jensen, Aurore, Massardier, Jérôme, Gauthier-Moulinier, Hélène, Gabor, Petra, Rahli, Djamila, Laurent, Juliette, Elaoun, Neila, Weil, Michèle, Hervé, François, Schnurgier, Aurélie, Leautez-Nainville, Sophie, Lamaury, Isabelle, Faye, Albert, Cazassus, François, Rajguru, Mandavi, Lagree, Marion, Burle, Christian, Cotte, Laurent, Dehlinger-Paul, Marion, Blum, Laurent, Joutel, Martine, Pommelet, Virginie, Perre, Philippe,, Ratsimbazafy, Lanto, Belgodere, Danièle, Simon-Toulza, Caroline, Vayssière, Christophe, Lotton, Pascal, Selleret, Lise, Fischer, Alain, Camus, Michel, Ben Salah, Mariam, Sibiude, Jeanne, Sow, Marie-Thérèse, Gromez, Alexis, Walter, Véronique, Truillet, Véronique, Marouts, Erianna Bellaton, Tabone, Marie-Dominique, Monpoux, Fabrice, Pathe, Jean-Paul, Philip, Gisèle, Braig, Suzanne, Blanche, Stephane, Chevojon, Pierre, Coursol, Anne, Michaud, Christophe, Caseris, Marion, Mesnard, Louis, Briandet, Claire, Ansart, Séverine, Entz-Werlé, Natacha, Houllier, Marie, Jault, Thierry, Yangui, Mohamed Amine, Lumbroso, Philippe, Tardif, Didier, Routier, Corinne, Goissen, Céline, Lesauder, Catherine, Ragnaud, Jean-Marie, Seaume, Hervé, Autret, Fanny, Neizelien, Joelle, Segondy, Michel, Chabrol, Amélie, Boutet, Arnaud, Bolot, Pascal, Marty, Laurence, Villemant, Agnès, Perre, Philippe, van De, Constanty, Anne, Demersay, Arnaud Chalvon, Costa, Myriam, Desmergers, Baya, Belloy, Marie, Delassus, Jean-Luc, Safwan, Hassan, Lavastre, Marie Laure, Moreau, Philippe, Bourgault, Olivier, David, Eric, Bounan, Stéphane, Werner, Evelyne, Blanc, Christine, Turquini, Marie-France, da Silva, Christelle Dusart, Murger, Patricia, Proust, Stéphanie, Horovitz, Jacques, Dina, Julia, Brochier, Corinne, Aubret, Valérie Raynal, Roux, Denis, Rudigoz, Rene-Charles, Mulard, Catherine, Weinbreck, Pierre, Mahlaoui, Nizar, Grand-Courault, Carole, Chirouze, Catherine, Granier, Michèle, Arvieux, Cédric, Bauville, Estelle, Galiba, Eliane, de Gennes, Christiane, Clavel, Cyril, Todorova, Darina, Moulin, Alice, Jeantils, Vincent, Hittinger, Gilles, Chabanier, Pierre, Veber, Florence, Pierronnet, Danielle, Valentin, Morgane, Bocket, Laurence, Tassi, Sylvie, Bonnenfant, Valerie, Clavere, Gaelle, Pinto-Cardoso, Gaelle, Courcoux, Mary-France, Boyer, Emeline, Habibi, Fakher, Vivier, Valérie, Balaz, Valérie, Maakroun, Zoha, May, Adrien, Boutaric, Emmanuelle, Pistone, Thierry, Rouha, Mahfoud, Messaoudi, Fabienne, Amel, Mahdi, Delveaux, Sandrine, Mazingue, Françoise, Jrad, Ikram, Taillet, Françoise, Pauly-Ravelly, Isolde, Tordjeman, Nathalie, Morau, Geneviève, Maurel, Elise, Favret, Véronique, Rehaiem, Sami, Elenga, Narcisse, Dienga, Etienne, Fischer, Patricia, Miantezila, Joe, Guimard, Karine, de Saint Martin, Luc, Deville, Anne, Kebaili, Kamila, Malet, Martine, Aubrard, Yves, Lupin, Catherine, Echard, Marie, Chamouilli, Jean-Marc, Driessen, Marine, Bry, Sandrine, Challier, Marion, Sanchez, Lydie, Labaune, Jean-Marc, Couderc, Sophie, Proust, Aurélie, Abdelhadi, Mohamed, Belkacem, Touria, Azria, Elie, Calvez, Christian, Mandelbrot, Laurent +416 morecore +1 more sourcePharmacokinetics and Drug–Drug Interactions of Long-Acting Intramuscular Cabotegravir and Rilpivirine
, 2021 Combined antiretroviral treatments have significantly improved the morbidity and mortality related to HIV infection, thus transforming HIV infection into a chronic disease; however, the efficacy of antiretroviral treatments is highly dependent on the ...Marzolini, C., Marzolini, C, Hodge, D, Back, DJ, Gibbons, S., Khoo, S.H., Khoo, SH, Back, D.J., Hodge, D., Gibbons, S +9 morecore +1 more sourcePharmacokinetics of Rilpivirine in HIV-Infected Pregnant Women [PDF]
, 2016 BACKGROUND: Rilpivirine pharmacokinetics is defined by its absorption, distribution, metabolism, and excretion. Pregnancy can affect these factors by changes in cardiac output, protein binding, volume of distribution, and cytochrome P450 (CYP) 3A4 ...Smith, Elizabeth, Tran, Anna H, Wang, Jiajia, George, Kathleen, Tran, Anna Hoang, Kreitchmann, Regis, Best, Brookie M, Cressey, Tim R, Rungruengthanakit, Kittipong, Capparelli, Edmund V, Chakhtoura, Nahida, Stek, Alice, Mirochnick, Mark, Burchett, Sandra K, Shapiro, David E +14 morecore +1 more sourceUse of PCR Signal and Therapeutic Drug Monitoring in a Switch Cohort Study to Tenofovir/Emtricitabine/Rilpivirine: A W96 Follow-Up. [PDF]
PLoS ONE, 2015 To assess, in a clinical cohort, the efficacy of switching treatment in virologically-suppressed patients to tenofovir/emtricitabine/rilpivirine as a single-tablet regimen (STR) using the PCR signal of the viral load (VL) assay and plasma drug ...Charlotte Charpentier, Minh Patrick Lê, Véronique Joly, Benoit Visseaux, Sylvie Lariven, Bao Phung, Patrick Yéni, Yazdan Yazdanpanah, Diane Descamps, Gilles Peytavin, Roland Landman +10 moredoaj +1 more source