Novel Sulfonylhydrazones With Sulfonate Ester Framework: Promising Dual Inhibitors of AChE and hCAs
ABSTRACT Alzheimer's disease (AD) is a progressive neurodegenerative disorder that affects millions of individuals worldwide. Treatment strategies for AD vary depending on cognitive and behavioral symptoms, with cholinergic replacement therapy using acetylcholinesterase (AChE) inhibitors being one of the primary approaches.
Cansu Öztürk +3 more
wiley +1 more source
This study investigated the anti‐inflammatory effects of 21α‐methylmelianol (MMN), a tirucallane triterpenoid isolated from Melia azedarach, in lipopolysaccharide‐ stimulated RAW264.7 macrophages in vitro, and in a dextran sodium sulfate‐induced ulcerative murine colitis model in vivo. ABSTRACT Melia azedarach L., also known as the chinaberry tree, has
Fan Cao +8 more
wiley +1 more source
Synthesis, physico-chemical and antimicrobial evaluation of Co(II) and Ni(II) complexes with Schiff base derived from sulphanilamine and salicylaldehyde [PDF]
Schiff base derived from sulphanilamine and salicylaldehyde was synthesized, its reaction with nickel(II) and cobalt(II) chloride in 2:1 mole ratio yielded Ni(II) and Co(II) complexes respectively.
Siraj, I.T., Yusuf, B.A.
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Laboratory classes in bioorganic chemistry [PDF]
биоорганическая химияЛабораторные занятия предназначены для иностранных студентов и включают 18 ...
Hidranovich, L. G., Khodos, O. A.
core
Ionizing Radiation Used in Drug Sterilization, Characterization of Radical Intermediates by Electron Spin Resonance (ESR) Analyses [PDF]
In this study, the feasibility of radiation sterilization of drugs/drug raw materials is investigated by using Electron Spin Resonance (ESR) spectroscopy.
Çolak, Şeyda
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AIM. To comparatively analyze thyroid abnormalities in patients with type 2 diabetes mellitus (DM2) in the past 10 years. MATERIALS AND METHODS. The thyroid state 10 years ago and presently was evaluated in 166 and 101 patient with DM2, respectively. The
I V Tereshchenko, A A Suslina
doaj
Toxicity of sulfanilamide in vitamins A and E deficient rabbits [PDF]
Digitized by Kansas State University ...
Kosuri, Narayana Rao
core
MODELING OF CARBONIC ANHYDRASE (II) INHIBITORY ACTIVITIES OF SULPHONILAMIDE SCHIFF BASES BY ARTIFICIAL NEURAL NETWORK TRAINED WITH DIFFERENT NUMERICAL TECHNIQUES [PDF]
Objective: The aim of the present study was to develop robust linear and non-linear Quantitative Structure-Activity Relationship (QSAR) models for exploring the relationship between the structural features of a series of sulphanilamide Schiff bases and ...
Pandey, Vandana
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Risk assessment of manufacturing and usage of test systems for quality control of compounded preparations [PDF]
Introduction: The development and implementation of test systems in pharmacy practice could be one of the ways of optimization of the quality control of compounded preparations. Test kits, which have been manufactured in a pharmacy, are simple, cheap and
Georgiyants, Viktoria +2 more
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Determination and evaluation of acidity constants of some imidazole and thiazole linked acetamide compounds [PDF]
In this work, the effect of substituents on the acidity constants of some acetamide derivatives was investigated. The acidity constants of nine acetamide derivatives were determined at 25 °C using a UV spectrophotometric method.
Demirayak, Şeref +3 more
core +1 more source

