Results 71 to 80 of about 90,509 (255)

Design and Synthesis of New N-(5-Trifluoromethyl)-1H-1,2,4-triazol-3-yl Benzenesulfonamides as Possible Antimalarial Prototypes

Molecules, 2011
A rational approach was used to synthesize a new set of 15 1H-1,2,4-triazol-3-yl benzenesulfonamide derivatives with the aim of developing new antimalarial lead compounds.
Nubia Boechat, Osvaldo A. Santos-Filho, Isabor C. Silva, Luiz C.S. Pinheiro   +3 more
doaj   +1 more source

Effect of Pyrolysis on the Removal of Antibiotic Resistance Genes and Class I Integrons from Municipal Wastewater Biosolids [PDF]

, 2018
Wastewater biosolids represent a significant reservoir of antibiotic resistance genes (ARGs). While current biosolids treatment technologies can reduce ARG levels in residual wastewater biosolids, observed removal rates vary substantially.
Kappell, Anthony D., Kimbell, Lee, McNamara, Patrick J.   +2 more
core   +1 more source

Discovery of macrocyclic inhibitors of apurinic/apyrimidinic endonuclease 1 [PDF]

, 2019
Apurinic/apyrimidinic endonuclease 1 (APE1) is an essential base excision repair enzyme that is upregulated in a number of cancers, contributes to resistance of tumors treated with DNA-alkylating or -oxidizing agents, and has recently been identified as ...
Beglov, Dmitri, Brown, Lauren E., Chen, Qiujia, Chennamadhavuni, Spandan, Georgiadis, Millie M., He, Hongzhen, Kelley, Mark R., Panek, James S., Porco, John A., Reed, April, Trilles, Richard, Vajda, Sandor, Wireman, Randall   +12 more
core   +7 more sources

Cycloauration of pyridyl sulphonamides [PDF]

, 2008
The pyridyl-2-alkylsulfonamides C₅H₄N(CH₂)nNHSO₂R (n = 1,2; R = Me, Ph or p-C₆H₄Me) and 8-(p-tosylamino)quinoline undergo facile cycloauration reactions with H[AuCl₄] in water, giving metallacyclic complexes coordinated through the pyridyl (or quinolyl ...
Henderson, William, Kilpin, Kelly Joan, Nicholson, Brian K.   +2 more
core   +2 more sources

An iron-chelating sulfonamide identified from Drosophila-based screening for antipathogenic discovery

, 2022
Yeon-Ji Yoo, In-Young Chung, Shivakumar S. Jalde, Hyun‐Kyung Choi, You‐Hee Cho   +4 more
openalex   +1 more source

Determination of quinolones and sulfonamides residues in aquatic products and livestock products with enhanced matrix removal-lipid adsorbent by liquid chromatography-tandem mass spectrometry

Shipin yu jixie
ObjectiveTo establish a new method for simultaneous detection of quinolones (QNs) and sulfonamides (SAs) in aquatic products and livestock products.MethodsIn pretreatment, this work compares the effect of extraction solvents on the recoveries and ...
QIN Yu, XUE Feng, YU Junjie, LIU Yang, GONG Heng   +4 more
doaj   +1 more source

Carbonic Anhydrase Inhibitors: Synthesis and Inhibition Against Isozymes I, II and IV of Topically Acting Antiglaucoma Sulfonamides Incorporatingcis-5-Norbornene-endo-3-Carboxy-2-Carboxamido Moieties [PDF]

, 2001
Angela Casini, Francesco Mincione, Marc A. Ilies, Luca Menabuoni, Andrea Scozzafava, Claudiu T. Supuran   +5 more
openalex   +1 more source

Design and Synthesis of Dy₂TmSbO₇/BiHoO₃ Heterojunction: The Mechanism and Application for Photocatalytic Degradation of Sulphamethoxypyridazine

Molecules
A novel Z-scheme Dy2TmSbO7/BiHoO3 heterostructure photocatalyst was synthesized with the ultrasound-assisted solvothermal method. The Dy2TmSbO7/BiHoO3 heterojunction photocatalyst (DBHP) reflected wonderful separation efficiency of photogenerated ...
Jingfei Luan, Minghe Ma, Liang Hao, Hengchang Zeng, Anan Liu   +4 more
doaj   +1 more source

In vivo Anti Inflammation Studies of Novel 1, 2, 5 Oxadiazole Sulfonamide Hybrids [PDF]

, 2021
Hafiz Adnan Ahmad, Muhammad Rahil Aslam, Salman Gul, Tariq Mehmood, Munawar Ali Munawar   +4 more
openalex   +1 more source

Crystal structure of potassium [4-amino-5-(benzo[d]thiazol-2-yl)-6-(methylsulfanyl)pyrimidin-2-yl](phenylsulfonyl)azanide dimethylformamide monosolvate hemihydrate

Acta Crystallographica Section E: Crystallographic Communications, 2019
The title compound, K+·C18H14N5O2S3−·C3H7NO·0.5H2O, was obtained in a reaction designed to deliver a neutral 2-pyrimidylbenzothiazole. The anion is deprotonated at the sulfonamide nitrogen. The asymmetric unit of the title compound contains two potassium
Rasha A. Azzam, Galal H. Elgemeie, Rokia R. Osman, Peter G. Jones   +3 more
doaj   +1 more source