Results 161 to 170 of about 9,794 (211)

The Thiazole Aldehyde Synthesis

Synthesis, 1998
Aldehydes with diverse structural arrays are prepared by construction of carbon chains at C-2 of the thiazole ring and conversion of the heterocycle into the formyl group. Various methods are described that differ depending on the type of thiazole-based reagent employed in the initial carbon-carbon bond forming reaction leading to 2-substituted ...
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Direct Arylation of Thiazoles on Water

Angewandte Chemie, 2007
Wetter is better: The direct arylation of thiazoles on water is quicker, cleaner, and higher-yielding than arylation in organic solvents. The reaction works under mild conditions for an array of aryl iodides, producing 2,5-diaryl thiazoles in excellent yields.
Turner, Gemma L., Morris, James A., Greaney, Michael F.   +2 more
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Imidazole, oxazole and thiazole alkaloids

Natural Product Reports, 2006
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
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Synthesis of Oligonucleotides Containing Thiazole and Thiazole N-Oxide Nucleobases

Organic Letters, 2002
[reaction: see text] The thiazole C-nucleoside analogue was synthesized by the Hantzsch cyclization method to form the thiazole ring and was then converted to the thiazole N-oxide C-nucleoside analogue by peracid oxidation of the heterocycle nitrogen.
Tod J, Miller, Hannah D, Farquar, Arsham, Sheybani, Camille E, Tallini, Andrea S, Saurage, Frank R, Fronczek, Robert P, Hammer   +6 more
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Thiazole Derivatives as Potential Chemotherapeutic Agents: Homolytic Arylation of Thiazole with Phenylazotriphenylmethane

Journal of Pharmaceutical Sciences, 1978
The homolytic arylation of thiazole with phenylazotriphenylmethane (as a free radical source) was carried out to explore the potential chemotherapeutic activity of the resulting triphenylmethyl derivatives. The experimental data differed from similar results on other isosteric heterocycles: one compound only was obtained, having both phenyl and ...
G, Fenech, A, Chimirri, R, Ficarra
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Thiazoles

2022
Agata Chotera-Ouda, Aneta Wróblewska, Paweł Tokarz, Christian V. Stevens   +3 more
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Thiazoles and Benzothiazoles

2012
This chapter highlights the recent developments in the metalation of thiazoles and benzothiazoles as well as the reactions of the resulting metalated species (2000 to present). Metalation reactions consist of lithiation (including halogen dance reactions), magnesation, zincation, caldation, boronation, and silylation, while application of the metalated
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Thiazolation of phenylthiosemicarbazone to access new thiazoles: anticancer activity and molecular docking

Future Medicinal Chemistry
Aim: Novel thiazole hybrids were synthesized via thiazolation of 4-phenylthiosemicarbazone (4). Materials & methods: The anticancer activity against the NCI 60 cancer cell line panel. Results: Methyl 2-(2-((1-(naphthalen-2-yl)ethylidene)hydrazineylidene)-4-oxo-3-phenylthiazolidin-5-ylidene)acetate (6a) showed significant anticancer activity at 10 μM ...
Walid E Elgammal, Safaa S Shaban, Essam M Eliwa, Ahmed H Halawa, Shimaa M Abd El-Gilil, Rasha A Hassan, Amr M Abdou, Gameel AM Elhagali, MAM Abdel Reheim   +8 more
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Synthesis of Thiazoles from Metalated Thiazoles

2010
P. A. Koutentis, H. A. Ioannidou
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Halogenation of Thiazoles and Thiazole 3-Oxides

2002
D. Kikelj, U. Urleb
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