Results 131 to 140 of about 2,743 (163)

Tautomeric Modification of GlcNAc-Thiazoline

Organic Letters, 2007
The potent O-GlcNAcase (OGA) inhibitor GlcNAc-thiazoline has been modified by buffer- or acylation-induced imine-to-enamine conversion and then electrophile or radical addition (Xn = D3, F, N3, OH, SMe, COCF3, CF3). Several functionalized GlcNAc-thiazolines show highly selective inhibition of OGA vs human hexosaminidase and thus have promise as tools ...
Spencer, Knapp, Mohannad, Abdo, Kehinde, Ajayi, Richard A, Huhn, Thomas J, Emge, Eun Ju, Kim, John A, Hanover   +6 more
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2‐Acetonyl‐thiazolin

Chemische Berichte, 1953
AbstractAus 2‐Methyl‐thiazolin und Keten wird 2‐Acetonyl‐thiazolin erhalten, das mit Kupfersalzen eine Komplex‐Verbindung liefert und im Rattenschwanz‐Test blutdrucksenkend wirkt.
Richard Kuhn, Günter Quadbeck, Erich Röhm   +2 more
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ChemInform Abstract: δ3‐Thiazolines, δ4‐Thiazolines, and Thiazoles from Penem Antibiotics.

ChemInform, 1992
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
G. VISENTIN, E. PERRONE, D. BORGHI, V. RIZZO, M. ALPEGIANI, A. BEDESCHI, R. CORIGLI, G. RIVOLA, G. FRANCESCHI   +8 more
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Synthesis and antioxidant activity of pyrazolyl-oxazolines/thiazolines and isoxazolyl-oxazolines/thiazolines

Medicinal Chemistry Research, 2013
A new class of pyrazolyl/isoxazolyl-oxazolines and thiazolines were synthesized from E-arylsulfonylethenesulfonylacetic acid methyl ester and tested for antioxidant activity. Among the tested compounds, 14b exhibited excellent antioxidant activity when compared with the standard ascorbic acid.
Adivireddy Padmaja, Chittoor Rajasekhar, Suram Durgamma, Bhumireddy Chinnachennaiahgari Venkatesh, Venkatapuram Padmavathi   +4 more
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Oligo‐(thiazolin)‐Naturstoffsynthese

Nachrichten aus Chemie, Technik und Laboratorium, 1995
Abstract“Synthese im Blickpunkt” will zur Beschäftigung mit neuen synthetischen Verfahren oder besonders eleganten und wichtigen Synthesen aus der aktuellen chemischen Literatur anregen ‐ ohne Anspruch auf Vollständigkeit. Die Rubrik erscheint alle zwei Monate und wird 1995 von Dr. Ulrich Koert, Universität Marburg, betreut.
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2‐Amino‐2‐thiazoline. V. phenylthioureido and phenylureido derivatives of 2‐thiazoline

Journal of Heterocyclic Chemistry, 1968
AbstractThe reaction of 2‐amino‐2‐thiazoline (I) with phenylisothiocyanate has been reported to give 2‐imino‐3‐phenylthiocarbamoylthiazolidine (II) at low temperatures and l‐phenyl‐3‐(2‐thiazolin‐2‐yl)‐2‐thiourea (III) at ca. 100°. When performed by us, however, this reaction gave only a single mono‐adduct regardless of the temperature.
Daniel L. Klayman, James J. Maul, George W. A. Milne   +2 more
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Synthesis of thiazolines and thiazolidines

Chemistry of Heterocyclic Compounds, 1972
Primary α-ethynylamines form thiazolines with isothiocyanates, while secondary α-ethynylamines give thiazolidines. Data on the IR, PMR, and UV spectra of the compounds obtained are presented.
I. N. Azerbaev, L. T. Kalkabaeva, M. Zh. Aitkhozhaeva, L. A. Tsoi   +3 more
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2-Methyl-2-thiazoline

2001
[2346-00-1] C4H7NS (MW 101.19) InChI = 1S/C4H7NS/c1-4-5-2-3-6-4/h2-3H2,1H3 InChIKey = JUIQOABNSLTJSW-UHFFFAOYSA-N (lithiation produces an acetaldehyde enolate equivalent for synthesis of mono-, di-, and trisubstituted acetaldehydes,1, 2 β-hydroxy aldehydes,3 homoallylic alcohols,3 and α,α-disubstituted β-ethylenic methyl ...
Todd D. Nelson, Albert I. Meyers
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Novel synthesis of 2-thiazolines

Tetrahedron Letters, 2000
Abstract The synthesis of a series of 2-thiazolines was carried out under mild conditions from the corresponding thiazolidines, by a Ru-catalyzed/TBHP oxidation reaction conditions. The reaction was chemoselective towards the amine-imine oxidation and was also regioselective, affording the unsaturation at the 2-position of the heterocycle, even with ...
Xavier Fernandez, Roland Fellous, Elisabet Duñach   +2 more
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Some Conversions of Thiazoline Carboxylic Acid Esters.

ChemInform, 2003
We have carried out solvolysis of the previously described ethyl esters of 3-methyl(aryl)-4-methyl-2-thioxothiazoline-5-carboxylic acids, leading to the corresponding acids without breaking down the heterocycle. We synthesized a series of novel esters from the latter by treatment with dimethyl sulfate or reactive halides.
V. V. Dovlatyan, K. A. Eliazyan, V. A. Pivazyan, A. P. Engoyan   +3 more
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