Results 181 to 190 of about 10,094 (251)

2-Oxoindolin-thiazoline hybrids as scaffold-based therapeutics for T2DM-associated cognitive impairment: design, synthesis, <i>in vitro</i> and <i>in silico</i> studies. [PDF]

RSC Med Chem
Qayed WS, Hassan MA, Şenol H, Taslimi P, Aboul-Fadl T.   +4 more
europepmc   +1 more source

Synthesis, Glucosidase Inhibition, and In Silico Modeling Analysis of Highly Fluorinated 2-Imino-1,3-thiazolines in Search of Potent Antidiabetic Agents. [PDF]

ACS Omega
Zahid LU, Zaib S, Saeed A, Alharbi HY, Aljohani MS, Alharbi O, Rana N, Khan I, Shabir G, Ahmed A, Saleem A, Awwad NS, Ibrahium HA.   +12 more
europepmc   +1 more source

Evaluation of the Drug-Induced Liver Injury Potential of Saxagliptin through Reactive Metabolite Identification in Rats. [PDF]

Pharmaceutics
Kim KY, Jeong YJ, Park SY, Park EJ, Jeon JH, Song IS, Liu KH.   +6 more
europepmc   +1 more source

Electrochemical aptasensor for 2-amino-2-thiazoline-4-carboxylic acid (ATCA), a metabolite for cyanide poisoning. [PDF]

Sci Rep
Khan HMA, Yusof NA, Ahmad SAA, Yu CY, Raston NHA, Rahman SFA.   +5 more
europepmc   +1 more source

An Efficient and Accessible Hectogram-Scale Synthesis for the Selective O-GlcNAcase Inhibitor Thiamet-G. [PDF]

ACS Omega
Holicek V, Deen M, Bhosale S, Ashmus RA, Vocadlo DJ.   +4 more
europepmc   +1 more source

Some of the next articles are maybe not open access.

Related searches:

New thiophene, thienopyridine and thiazoline-based derivatives: Design, synthesis and biological evaluation as antiproliferative agents and multitargeting kinase inhibitors.

Bioorganic chemistry (Print), 2022
Multitargeting kinase inhibitors recently proved to be a profitable approach for conquering cancer proliferation. The current study represents the design and synthesis of new thiophene, thienopyridine, and thiazoline-based derivatives 4-14a,b.
Zahra M. Alamshany, N. Tashkandi, Ismail M. M. Othman, M. Anwar, E. Nossier   +4 more
semanticscholar   +1 more source

A NIR fluorescent sensor based on thiazoline-isophorone with low cytotoxicity in living cells for Hg2+ detection through ICT associated hydrogen bonding effect.

Analytica Chimica Acta, 2021
Mercury (Hg) is a toxic pollutant and may cause serious health and environmental threats even at low concentrations. Thus, sensitive, efficient, and accurate techniques for the detection of Hg2+ ions in biological systems are in particular demand. In the
Serkan Erdemir, Mehmet Oguz, S. Malkondu
semanticscholar   +1 more source

2-thiazoline-2-thiol functionalized gold nanoparticles for detection of heavy metals, Hg(II) and Pb(II) and probing their competitive surface reactivity: A colorimetric, surface enhanced Raman scattering (SERS) and x-ray photoelectron spectroscopic (XPS) study

, 2021
A novel 2-thiazoline-2-thiol functionalized gold (Au-TT) nanosensor was developed for the selective and sensitive detection of toxic heavy metal ions, Hg(II) and Pb(II) by colorimetry, and for studying its competitive surface reactivity using SERS and ...
Ridhima Chadha, Abhishek Das, Anil K. Debnath, S. Kapoor, N. Maiti   +4 more
semanticscholar   +1 more source

Design, synthesis, X-ray analysis, and biological screening of new oxime and enaminone thiazoline-2-thione derivatives

, 2021
An urgent need exists to develop antimicrobial and anticancer drugs that are safer and less prone to the development of resistance. To this end, a series of 12 new thiazoline-2-thione derivatives (oxime and enaminone) were synthesized using an ...
Y. Asiri, A. Muhsinah, Abdulrhman Alsayari, H. Ghabbour, Z. Almarhoon, Faiz A. Al-aizari, K. Venkatesan, S. Tasqeeruddin, Syeda Shaheen Sulthana, Y. Mabkhot   +9 more
semanticscholar   +1 more source

Novel thiazoline-phenothiazine based “push-pull” molecules as fluorescent probes for volatile acids detection

, 2020
A series of novel acceptor-donor-acceptor type of “push-pull” molecules 3a-3e containing acid-sensitive component based on phenothiazine-5-oxide and thiazoline as donor and acceptor units, respectively were synthesized in excellent yields of 84–95 %. The
S. Chaudhary, Madhubani Mukherjee, T. Paul, S. Taraphder, M. Milton   +4 more
semanticscholar   +1 more source