Results 21 to 30 of about 2,667 (235)

The fluorescence‐based competitive counterflow assay developed for organic anion transporting polypeptides 1A2, 1B1, 1B3 and 2B1 identifies pentamidine as a selective OATP1A2 substrate

open access: yesThe FASEB Journal, Volume 37, Issue 11, November 2023., 2023
The fluorescent competitive counterflow assay can distinguish between substrates and non‐transported inhibitors of Organic anion transporting polypeptides. Substrates trigger efflux or the fluorescent probe from the cells. With this method, we identify the FDA‐approved antiprotozoal drug pentamidine as a selective OATP1A2 substrate. OATP1A2 can mediate
Orsolya Ungvári   +3 more
wiley   +1 more source

Discovery of Antitrypanosomal Indolylacetamides by a Deconstruction–Optimization Strategy Applied to Paullones

open access: yesChemMedChem, Volume 18, Issue 10, May 16, 2023., 2023
Treatment of Chagas disease, African sleeping sickness and Leishmaniasis is currently limited to few, unfavorable drugs. We discovered novel antitrypanosomal compounds via molecular simplification of an original molecule (MOL2008) displaying limited selectivity.
Jens C. Lindhof   +9 more
wiley   +1 more source

Prevalência de Tripanosoma vivax em bovinos no município de Patos de Minas/MG

open access: diamondRevista Acadêmica: Ciência Animal, 2017
Pedro Henrique Vieira Germano et al.
openaire   +3 more sources

Trypanosoma sp. em jacaré, Caiman crocodilus yacare (Daudín, 1823) (Crocodilia: Alligatoridae)

open access: yesSemina: Ciências Agrárias, 1990
Infecção natural por Trypanosoma sp. é descrita em jacaré, Caiman crododilus yacare (Crocodilia: Alligatoridae) em Mato Grosso do Sul, Brasil. O tripanosoma distingue-se de Trypanosoma grayi, do crocodilo Africano, Crocodilus niloticus (Crocodilia ...
Vânia Lúcia Brandão Nunes   +1 more
doaj   +1 more source

Trypanosoma (Megatrypanum shawi n. sp., um parasita de capivara, Hydrochaeris hydrochaeris (Linnaeus, 1766) (Rodentia: hydrochoeridae)

open access: yesSemina: Ciências Agrárias, 1987
Trypanosoma (Megatrypanum) shawi, n.sp., é descrito em capivara, Hydrochaeris hydrochaeris, no estado de Mato Grosso do Sul, Brasil. Os animais examinados apresentavam aspecto saudável e as parasitemias eram extremamente baixas.
Vânia Lúcia Brandão Nunes   +4 more
doaj   +1 more source

Nota sobre a infecção de Lutzomyia evandroi (Diptera: Psychodidae) por Ascocystis chagasi (Adler & Mayrink, 1961) no Estado do Maranhão Infection of Lutzomyia evandroi (Diptera: Psychodidae) by Ascocystis chagasi (Adler & Mayrink, 1961) in the State of Maranhao

open access: yesMemorias do Instituto Oswaldo Cruz, 1984
Encontramos a gregarina Ascocystis chagasi, bem como um nematódeo e um tripanosoma nao identificados, em Lutzomyia evandroi da ilha de São Luis, Maranhão.The gregarine Ascocystis chagasi as well as a nematode and an unidentified Trypanosome were found in
Reginaldo Peçanha Brazil, Lee Ryan
doaj   +1 more source

Reduction and Preparation of a Phthalimide Derivative from a Furo-heliangolide

open access: yesMolecules, 2000
Goyazensolide, a biologically active natural product classified as a furoheliangolide, was transformed in a phthalimide derivative that showed an enhanced biological activity against Tripanosoma cruzi.
Mauricio Gomes Constantino   +2 more
doaj   +1 more source

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