Results 141 to 150 of about 11,638,573 (298)

Discovery of new Schiff bases of the disalicylic acid scaffold as DNA gyrase and topoisomerase IV inhibitors endowed with antibacterial properties [PDF]

DNA gyrase and topoisomerase IV show great potential as targets for antibacterial medicines. In recent decades, various categories of small molecule inhibitors have been identified; however, none have been effective in the market. For the
Abou-Zied, Hesham A., Al-Wahaibi, Lamya H., Alzahrani, Hayat Ali, Bräse, Stefan, Gomaa, Hesham A. M., Mahmoud, Mohamed A., Rabea, Safwat M., Youssif, Bahaa G. M.   +7 more
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Synthesis and Study of Some 4-Chlorophenoxy Methyl Substituted amido1,3,4-Oxadiazoles, 1,3,4-Thiadiazoles and 1,2,4-Triazoles from 4-Chloro phenoxy acetic acid [PDF]

, 2013
Mudhar A. Othman, Khalid M. Daoud
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Novel quinazolin-4(3H)-one bionic-alkaloids bearing an 1,3,4-oxadiazole fragment as potential fungicides inhibiting Botrytis cinerea: Design, synthesis and bioactive-guided structural optimization

, 2023
Xiaobin Wang, Lili Yan, Juan Zhang, Yilin Zhang, Zongqun Zhang, Quanqing Zhao, Qingfang Cheng, Weihua Zhang   +7 more
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Synthesis and Antibacterial Activity of Some Novel Schiff S-Bases Compounds Containing Oxadiazole Ring

Ibn Al-Haitham Journal for Pure and Applied Sciences, 2019
Condensation of 4-methoxybenzoyl hydrazine with 4- aminobenzoic acid in the presence of POCl3 gave the oxadiazole derivative [III] .This compound was demethylated with aluminium chloride to give series of 2- (4-hydroxy phenyl)-5-(4-amino phenyl) 1,3 ...
J. H. Tomma, A. H. Raheema, I. H. Rouil
doaj  

Sensitization of an oxadiazole derivative as an organic photoconductor [PDF]

, 1982
The sensitization and the spectral sensitization of the photoconductivity of an organic derivative, 2,5-bis (p-diethyl-aminophenyl) - 1,3, 4-oxadiazole, was studied once an electrostatic sensitometer had been built.
Ceintrey, Claude G.
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Synthesis OF Ligands O.F BIS-Oxadiazole Triazole Witb Open OR Close Sides and Their Complxes With (Ctlf, Pdll) -

Ibn Al-Haitham Journal for Pure and Applied Sciences, 2017
A  OUI,tiper  of LWW lig_;:tnds  .of  ppen sides. of Bis-'Oxad1azoJe· and· Bis-triazole   derived from dichloroetbane  and  [Bis  0-ohloro   et!:ty) = :=::                                                 = ether)] (BCEE)' wersynthesi:zed ...
W.K. Me.hdi, F. H. Musa, H. A. Fadhel
doaj  

Synthesis, enzyme kinetics and computational evaluation of N-(β-d-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors [PDF]

, 2017
Begum, Jaida, Docsa, Tibor, Gergely, Pál, Hayes, Joseph M., Juhász, László, Polyák, Mária, Somsák, László, Szilágyi, Bence, Varga, Gergely   +8 more
core   +1 more source

Synthesis of [¹⁸F] 4‐amino‐N‐(3‐chloro‐4‐fluorophenyl)‐N′‐hydroxy‐1,2,5‐oxadiazole‐3‐carboximidamide (IDO5L): a novel potential PET probe for imaging of IDO1 expression

, 2015
Xuan Huang, Robert J. Gillies, Haibin Tian   +2 more
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Synthesis of N‐[{5‐Aryl‐1,3,4‐oxadiazole‐2‐yl}methyl]‐4‐methoxyaniline Derivatives and Their Anticonvulsant Activity [PDF]

, 2013
Basavapatna N. Prasanna Kumar, K. N. Mohana, L. Mallesha   +2 more
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Synthesis, spectral analysis and biological evaluation of 2-{[(morpholin-4-yl)ethyl]thio}-5-phenyl/aryl-1,3,4-oxadiazole derivatives.

, 2021
Azizur Rehman, Samreen Gul Khan, Syed Ali Raza Naqvi, Matloob Ahmad, Naheed Akhtar, Tanveer Hussain Bokhari, Muhammad Irfan, Ali Usman, Sidra Batool, Shahid Rasool, Syed Adnan Alı Shah, Muhammad Shahid   +11 more
openalex   +1 more source