Results 141 to 150 of about 5,910 (205)

An Imidazo[2,1-b][1,3,4]thiadiazole Derivative Inhibits the Virulence Factor α-Hemolysin by Blocking the Pullout of Its Stem Domain. [PDF]

ChemMedChem
Korotkov VS, Lukat P, Di Lucrezia R, Shekhar A, Degenhart C, Diestel R, Bilitewski U, Dinkel K, Blankenfeldt W, Brönstrup M.   +9 more
europepmc   +1 more source

Influence of Available Hydrophobic Interactions in New 2‑(Propylthio)‑<i>N</i>‑(1,3,4-thiadiazol-2-yl)nicotinamide Pharmacophore and Evaluation of Its Therapeutic Potential. [PDF]

ACS Omega
Nachimuthu L, Desikan R.
europepmc   +1 more source

Design, synthesis and antiproliferative, apoptotic, and immunomodulatory properties of new heteroaryl pyridine-linked 1,2,4-oxadiazoles as prospective dual EGFR/BRAF^V600E inhibitors. [PDF]

RSC Adv
Gomaa HAM, Shaker ME, Alzarea SI, Alatwi E, Mohamed FAM, Abdullah Alzahrani AY, Alyami BA, Bräse S, Rabea SM, Youssif BGM.   +9 more
europepmc   +1 more source

Reaction of &alpha;-Bromoacetophenones with 2-Anino-1, 3, 4-thiadiazoles

YAKUGAKU ZASSHI, 1952
Taizo Matsukawa, Syoiti Ban
openaire   +2 more sources

Unanticipated Reactivity toward Nucleophilic Attack in the Synthesis of Saccharyl-1,3,4-Thiadiazolyl Conjugates: Structure and Mechanistic Insights. [PDF]

J Org Chem
Guerreiro BEC, Carvalho DF, Coelho JAS, Paixão JA, Frija LMT, Cristiano MLS.   +5 more
europepmc   +1 more source

Antimicrobial Activity of 1,3,4-Thiadiazole Derivatives. [PDF]

Pharmaceuticals (Basel)
Górecki S, Kudelko A, Olesiejuk M.
europepmc   +1 more source

An exploration of potent antileishmanial agents derived from quinoline-thiazole and thiadiazole hybrids, targeting DHFR-TS and PTR1: design, synthesis, and computational analyses. [PDF]

RSC Med Chem
Rashdan HRM, Bekhit AA, Furlan V, Amagase K, Elshamy AI, Elfar N, Abdo MR, Ibrahim TM, Bren U, Eldehna WM, Sabt A.   +10 more
europepmc   +1 more source

Spectroscopic and theoretical studies of fluorescence effects in 2-methylamino-5-(2,4-dihydroxyphenyl)-1,3,4-thiadiazole induced by molecular aggregation [PDF]

, 2017
Gagoś, Mariusz, Górecki, Andrzej, Kosztołowicz, Katarzyna, Makowski, Marcin, Matwijczuk, Arkadiusz, Niewiadomy, Andrzej, Skrzypek, Alicja, Waś-Mrozek, Joanna   +7 more
core   +1 more source

Advanced Spectroscopic Studies of the AIE-Enhanced ESIPT Effect in a Selected 1,3,4-Thiadiazole Derivative in Liposomal Systems with DPPC. [PDF]

Int J Mol Sci
Skrzypek A, Budziak-Wieczorek I, Ślusarczyk L, Górecki A, Kamiński D, Kwaśniewska A, Okoń S, Różyło I, Matwijczuk A.   +8 more
europepmc   +1 more source

Synthesis, molecular modeling and harnessing the antimicrobial activity of new pyrazine-thiadiazole hybrids. [PDF]

BMC Chem
Abumelha HM, Halawani NM, Alharbi AS, Alsulami RN, Qurban J, Alomari KB, Al-Bonayan AM, El-Metwaly N.   +7 more
europepmc   +1 more source