Synthesis and Antiviral Activity of 5‑(4‑Chlorophenyl)-1,3,4-Thiadiazole Sulfonamides [PDF]
Starting from 4-chlorobenzoic acid, 10 new 5-(4-chlorophenyl)-N-substituted-N-1,3,4-thiadiazole-2-sulfonamide derivatives were synthesized in six-steps. Esterification of 4-chlorobenzoic acid with methanol and subsequent hydrazination, salt formation and
Zhuo Chen, Weiming Xu, Song Yang
exaly +4 more sources
Synthesis and Evaluation of Antimicrobial Activity of 1, 3, 4-Thiadiazole Analogues for Potential Scaffold. [PDF]
Pathogenic microbes are causal agents for various types of severe and even lethal infectious diseases. Despite of development in medication, bacterial and fungal infections still persist to be a vital problem in health care. Bacteria and several fungal species have shown resistance to antibiotics used in treatment to current medications.
Sahu S, Sahu T, Kalyani G, Gidwani B.
europepmc +5 more sources
Benzo[1,2-d:4,5-d′]bis([1,2,3]thiadiazole)-4-carbonitrile [PDF]
Electron-withdrawing heterocyclic units are found in most organic optoelectronic materials. Benzo[1,2-d:4,5-d′]bis([1,2,3]thiadiazole) is an interesting new heterocyclic system, the chemical properties of which are much less studied than other fused ...
Timofey N. Chmovzh +3 more
doaj +2 more sources
Synthesis and Bioactivity Evaluation of Novel Thiochroman-4-One Derivatives Incorporating Carboxamide and 1, 3, 4-Thiadiazole Thioether Moieties [PDF]
A series of novel thiochroman-4-one derivatives incorporating carboxamide and 1, 3, 4-thiadiazole thioether moieties were synthesized. Bioassay results indicated that the EC50 values of compound 6-chloro-N-(5-(methylthio)-1, 3, 4-thiadiazol-2-yl)-4 ...
Lu Yu +5 more
doaj +2 more sources
Synthesized azodyes of 2-amino-1, 3, 4- thiadiazole - 5 - thiol
Several azo dyes were synthesized through coupling reaetion of some substituted phenols and B.naphthol with diazonium salt of 2- amino-1,3-4- thiadiazol -5- thiol. All the synthesized compounds during this work were characterized using some speetral data
Baghdad Science Journal
doaj +4 more sources
Synthesis, Characterization and Biological Activates Studies of some New Derivatives From 2-aminoo-5-mercapto-1, 3, 4-thiadiazole [PDF]
In this work, thiadiazole derivatives were prepared by taking advantage of active sites in (2-amino-5-mercapto-1, 3, 4-thiadiazole) as a starting material base.
Baghdad Science Journal
doaj +5 more sources
Water/Alkali-Catalyzed Reactions of Azides with 2‑Cyanothioacetamides. Eco-Friendly Synthesis of Monocyclic and Bicyclic 1,2,3-Thiadiazole-4-carbimidamides and 5‑Amino-1,2,3-triazole-4-carbothioamides [PDF]
The reactions of thioamides with azides in water were studied. It was reliably shown that the reaction of 2-cyanothioacetamides 1 with various types of azides 2 in water in the presence of alkali presents an efficient, general, one-step, atom-economic ...
Nikolai A. Beliaev (7461455) +9 more
core +7 more sources
Theoretical Study of Interaction Between Thiadiazole Derivatives on Fe(110) Surface [PDF]
The theoretical performance of 4-methoxyphenyl-1,3,4-thiadiazole (AMPT), 2-Amino-5-(4-chlorophenyl)-1,3,4-thiadiazole (ACPT) and 2-amino-5-phenyl-1,3,4-thiadiazole (APT) as inhibitors of iron corrosion was assessed with a view of determining the ...
Thomas Nyijime +3 more
doaj +1 more source
Ionic Liquid Catalyzed One-Pot Synthesis of 5-(4-Substituted-Phenyl)-1,3,4-Thiadiazole-2-Amines [PDF]
A highly efficient ionic liquid catalyzed protocol has been investigated for the synthesis of 5-(4-substituted-phenyl)-1,3,4-thiadiazole-2-amine derivatives from the cyclocondensation of diversely substituted aromatic carboxylic acid and ...
Dinesh Lingampalle (14277729) +3 more
core +1 more source
Thiadiazole-Derived Covalent Organic Framework Macroscopic Ultralight Aerogel [PDF]
Shaping covalent organic frameworks (COFs) into macroscopic objects for practical application remains a huge challenge. Herein, a new thiadiazole-derived COF macroscopic ultralight aerogel (NNS-VCOF) was prepared through acid-catalyzed aldol condensation
Haifeng Ji (780358) +8 more
core +7 more sources

