Results 41 to 50 of about 1,760 (172)

Effects of the 5-HT1A agonist (??)-8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) on cocaine choice in cynomolgus monkeys

, 2005
Drugs that alter brain serotonin (5-HT) function can modulate the behavioral effects of cocaine, but the underlying receptor mechanisms are poorly understood. The present study examined the effects of the selective 5-HT1A receptor agonist (+/-)-8-hydroxy-
Nader, M A, Czoty, PW, Czoty, P W, Mccabe, Ciara, Nader, MA, McCabe, C   +5 more
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Avaliação da participação do receptor 5-HT1A pós-sináptico na hipofagia induzida pela injeção de 8-OH-DPAT na área hipotalâmica lateral [PDF]

, 2012
Dissertação (mestrado) - Universidade Federal de Santa Catarina, Centro de Ciências Biológicas. Programa Multicêntrico de Pós-Graduação em Ciências FisiológicasEstudos conduzidos em nosso laboratório avaliaram os efeitos da injeção local de 8-hidroxi-2 ...
Lavado, Cristiane
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Mediation of the discriminative stimulus properties of 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT) by the putative 5-HT1A receptor

, 1987
Male Sprague-Dawley rats were trained to discriminate the putative 5-HT1A receptor agonist, 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT) from saline in a 2-lever operant drug discrimination paradigm.
Kidd, Emma Jane, Neill, J., Tricklebank, M. D., Fozard, J. R.   +3 more
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Further characterisation of [3H]8-hydroxy-2-(DI-Npropylamino)tetralin bynding sites in human brain postmortem.

, 1997
The saturation parameters and the pharmacological characteristics of the binding of the serotonin 1A (5-HT1A) receptor agonist [H-3]8-hydroxy-2-(di-N-propylamino)tetralin ([H-3]8-OH-DPAT), as well as the effects of nucleotides and divalent cations (Mg2+,
Marazziti D, Batistini A, BEVILACQUA, GENEROSO, Rotondo A, Cassano GB, Borsini F, PALEGO, LIONELLA, Ladinsky H, LUCACCHINI, ANTONIO, NACCARATO, ANTONIO GIUSEPPE   +9 more
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Efeitos do bloqueio de receptores a1 do núcleo mediano da rafe sobre o comportamento alimentar e expressão da proteína Fos [PDF]

, 2014
Tese (doutorado) - Universidade Federal de Santa Catarina, Centro de Ciências Biológicas, Programa de Pós-Graduação Multicêntrico em Ciências Fisiológicas, Florianópolis, 2014A serotonina (5HT) é um neurotransmissor envolvido no controle da ingestão de ...
Silva, Eduardo Simão da
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Alkaloids from Eschscholzia californica and Their Capacity to Inhibit Binding of [³H]8-Hydroxy-2-(di-N-propylamino)tetralin to 5-HT_1A Receptors in Vitro^#

, 2016
A 70% ethanol extract of California poppy (Eschscholzia californica) was able to bind to 5-HT1A and 5-HT7 receptors at 100 μg/mL. The subsequent isolation procedure yielded the known alkaloids californidine (1), escholtzine (2), N-methyllaurotetanine (3),
Megan M. McCollom (2646292), Stefan Gafner (1828096), Kerry L. McPhail (418940), Chantal Bergeron (317019), Fiona E. Russell (2646295), Birgit M. Dietz (433364), Jason W. Budzinski (2646298), Jan A. Glinski (2167159), Ian M. Scott (2257921), Brian C. Foster (130023), Judy L. Bolton (194650), Mee-Ra Rhyu (300475)   +11 more
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Differential regulation of somatodendritic serotonin 5-HT1A receptors by 2-week treatments with the selective agonists alnespirone (S-20499) and 8-hydroxy-2-(Di-n-propylamino)tetralin: microdialysis and autoradiographic studies in rat brain

, 1999
Single treatment with the serotonin (5-hydroxytryptamine) 5-HT1A receptor agonists 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) and alnespirone (S-20499) reduces the extracellular 5-HT concentration (5-HText) in the rat midbrain and forebrain ...
M. T. Vilaró, Artigas, Francesc, J. M. Casanovas, Mengod Los Arcos, Guadalupe, Casanovas, Josep M., F. Artigas, Vilaró, Maria Teresa, G. Mengod   +7 more
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Alterations of In-vitro 5-HT Receptor Pharmacology as a Function of Multiple Treatment with 5-Hydroxytryptamine or 8-Hydroxy-2-(di-N-propylamino) Tetralin in Rat Isolated Aorta, Uterus and Fundus, and Guinea-pig Isolated Trachea

, 1994
The effects of single and multiple (5, 10, or 15 days) administration of the 5-HT1A agonist 8-hydroxy-2-(di-N-propylamino) tetralin (8-OH-DPAT) (3 mg kg−1, i.p.) or 5-HT (3 mg kg−1, i.p.) in-vivo on the response of selected isolated smooth muscles to 5 ...
David R Helton, Walter E Colbert
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Effects of the dopamine D₃ receptor agonist 7-hydroxy-2-(di-N -propylamino) tetralin in hyperthyroidism-induced premature ejaculation rat model

, 2018
Various factors are involved in the aetiology of premature ejaculation (PE). Hyperthyroidism is one of the causes of acquired PE, but the exact mechanism by which it causes the disorder is not yet understood.
O. Cinar, Esen, AHMET ADİL, Gidener, S., Durmus, NERGİZ, S. Gidener, N. Durmus, O. Demir, Aslan, GÜVEN, A. S. Evcim, A. A. Esen, G. Aslan, Demir, O., Cinar, O., Evcim, A. S.   +13 more
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Assessment of cocaine-like discriminative stimulus effects of dopamine D3 receptor ligands

, 1995
The highly selective dopamine D-3 receptor ligand, (+)-PD 128907 4aR10bR-(+)-trans-3,4,4a,10b-tetrahydro-4-n-propyl- 2H5H[4,3-b]-1,4-oxazin-9-ol), and other dopamine D-3 receptor ligands, (+/-)-7-hydroxy-2-(N,N-di-n-propylamino)tetralin and (+)-7-hydroxy-
Geter-Douglass, B, Witkin, J M, Durk Dijkstra, Håkan Wikström, WITKIN, JM, Jane B. Acri, Carter, S R, Beth Geter-Douglass, ACRI, JB, GETERDOUGLASS, B, Ken Alling, Jonathan L. Katz, Jeffrey M. Witkin, Sean R. Carter, Katz, J L, Acri, J B, Alling, K, Wikstrom, H, Dijkstra, D, CARTER, [No Value], KATZ, JL   +20 more
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