Results 91 to 99 of about 989 (99)

Allosteric Integrase Inhibitors

2016
Victoria Hann, Peter Dawson, Mark Ashton
openaire   +1 more source

A Potent Allosteric Inhibitor of HIV-1 Integrase

Synfacts, 2022
openaire   +1 more source

Expeditious Synthesis of a Potent Allosteric HIV-1 Integrase Inhibitor GSK3839919A

Organic Process Research & Development, 2023
Mark A. Bobko, Jennifer M. Elward, B. Narasimhulu Naidu, Yexenia E. Nieves-Quinones, Christopher A. Reiher, Qiaogong Su, Liang Sun, John Woodard, Shiping Xie, Wuxing Yang, Yunxing Yin   +10 more
openaire   +1 more source

HIV-1 Integrase catalytic core domain complexed with allosteric inhibitor STP03-0404

, 2020
Jared Lindenberger, Mamuka Kvaratskhelia
openalex   +1 more source

HIV-1 Integrase Catalytic Core Domain Complexed with Allosteric Inhibitor (2S)-tert-butoxy[6-(5-chloro-1H-benzimidazol-2-yl)-2,5-dimethyl-4-phenylpyridin-3-yl]ethanoic acid

, 2014
Lili Feng, Mamuka Kvaratskhelia
openalex   +1 more source

HIV-1 Integrase Catalytic Core Domain Complexed with Allosteric Inhibitor (2S)-tert-butoxy[4-(4-chlorophenyl)-6-(3,4-dimethylphenyl)-2,5-dimethylpyridin-3-yl]ethanoic acid

, 2014
Lili Feng, Mamuka Kvaratskhelia
openalex   +1 more source

HIV-1 Integrase Catalytic Core Domain (CCD) in Complex with a Fragment-Derived Allosteric Inhibitor

, 2016
Dinshaw J. Patel, Joseph D. Bauman, Eddy Arnold   +2 more
openalex   +1 more source

Structural Impact of Ex Vivo Resistance Mutations on Hiv-1 Integrase Polymers Induced by Allosteric Inhibitors

Saira Montermoso, Grant Eilers, Audrey Allen, Robert Sharp, Young Sun Hwang, Frederic D. Bushman, Kushol Gupta, Gregory Van Duyne   +7 more
openalex   +1 more source

The LEDGINs: first-in-class allosteric HIV-1 integrase inhibitors with potential pre-clinical development

, 2011
Belete A. Desimmie, Frauke Christ, Arnout Voet, Arnaud Marchand, Stefan Nicolet, Damien Marchand, Sergei V. Strelkov, Marc De Maeyer, Patrick Chaltin, Zeger Debyser   +9 more
openalex