Results 311 to 320 of about 1,043,535 (340)
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Hormone and Metabolic Research, 1986
The three classes of CCK antagonists illustrate the various factors governing affinity of the antagonists for the CCK receptor. The major influence in determining potency of the cyclic nucleotide derivatives, amino acid derivatives and C-terminal fragments of CCK, are hydrophobic forces.
P N, Maton, R T, Jensen, J D, Gardner
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The three classes of CCK antagonists illustrate the various factors governing affinity of the antagonists for the CCK receptor. The major influence in determining potency of the cyclic nucleotide derivatives, amino acid derivatives and C-terminal fragments of CCK, are hydrophobic forces.
P N, Maton, R T, Jensen, J D, Gardner
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2007
Androgens are essential for the development and maintenance of male sexual characteristics. They exert their effects through the androgen receptor, which is a member of the …
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Androgens are essential for the development and maintenance of male sexual characteristics. They exert their effects through the androgen receptor, which is a member of the …
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Nature, 1969
IF drugs b and c are competitive antagonists of drug a, then it would seem self evident that the addition of c to a system in which b was already present would increase the degree of block. But where the receptors are exposed to the agonist for only a short time there is another possibility. If the first antagonist dissociates from the receptors slowly,
R P, Stephenson, B L, Ginsborg
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IF drugs b and c are competitive antagonists of drug a, then it would seem self evident that the addition of c to a system in which b was already present would increase the degree of block. But where the receptors are exposed to the agonist for only a short time there is another possibility. If the first antagonist dissociates from the receptors slowly,
R P, Stephenson, B L, Ginsborg
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Australian and New Zealand Journal of Medicine, 1984
The realisation that serotonin plays a role not only in the carcinoid syndrome but also in migraine, nociception, dumping syndrome, vascular disease and hypertension, has led to an enormous amount of activity in search of serotonin antagonists. Numerous such pharmacological agents have been identified but only few have found their way into clinical use.
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The realisation that serotonin plays a role not only in the carcinoid syndrome but also in migraine, nociception, dumping syndrome, vascular disease and hypertension, has led to an enormous amount of activity in search of serotonin antagonists. Numerous such pharmacological agents have been identified but only few have found their way into clinical use.
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2013
Kisspeptin is now known to be an important regulator of the hypothalamic--pituitary-gonadal axis and is the target of a range of regulators, such as steroid hormone feedback, nutritional and metabolic regulation. Kisspeptin binds to its cognate receptor, KISS1R (also called GPR54), on GnRH neurons and stimulates their activity, which in turn provides ...
Antonia Kathryn, Roseweir +1 more
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Kisspeptin is now known to be an important regulator of the hypothalamic--pituitary-gonadal axis and is the target of a range of regulators, such as steroid hormone feedback, nutritional and metabolic regulation. Kisspeptin binds to its cognate receptor, KISS1R (also called GPR54), on GnRH neurons and stimulates their activity, which in turn provides ...
Antonia Kathryn, Roseweir +1 more
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Antagonists to the benzodiazepines
British Dental Journal, 1984P, McGonigal, C N, Schofield
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