Antifertility and Antiproteolytic Activity of Activated N‐Carbobenzoxy Amino Acid Esters
Journal of Pharmaceutical Sciences, 1979N-Carbobenzoxy L-phenylalanine, glycine, L-leucine, and L-proline derivatives, their vinyl esters, and their 1,2-dibromoethyl esters were tested for antifertility activity in mice. Intraperitoneal administration reduced the pregnancy percentage and the number of fetuses per litter.
I H Hall, Larry J Loeffler
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Influence of Sex and Thyroid Principles on the Antiproteolytic Activity of Rat Serum
Thrombosis and Haemostasis, 1966SummaryExamination of antiproteolytic activity in rats administered sex steroids and thyroid principles revealed the following :Female rats display lower serum antitrypsin and antiplasmin activity than their male counterpart under all conditions investigated.
C I, Wabner, J L, Gray, W F, Blatt
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Aromatic tetra-amidines with antiproteolytic activity inhibit platelet aggregation and secretion
Thrombosis Research, 1989We have investigated the possibility that TAPP-H may control platelet aggregation and serotonin release induced by a series of physiological and non-physiological stimuli, that are selected on the ground of their molecular mechanism. The search of new antiplatelet molecules may have relevant implications in the therapy of haemostasis ...
Roberto Ferroni, Serena Traniello
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ON THE ANTITHROMBIC AND ANTIPROTEOLYTIC ACTIVITY OF ALPHA TOCOPHERYL PHOSPHATE
American Journal of Physiology, 1948K L Zierler
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Study of the Antiproteolytic Activity of Fenamates and Indomethacin
Pharmacology, 1973The effect of mefenamic acid, flufenamic acid and of indomethacin on tryptic hydrolysis of bovine albumin (BA) and of the syn thetic substrates N-benzoyl-DL.-arginine-p-nitro anilide (BAPNA) and L-lysin-p-nitroanilide (LPA) was studied in vitro. Both fenamates and indomethacin inhibited tryptic hydrolysis of BA, indomethacin being more active.
M, Stanciková, K, Trnavský
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Antiproteolytic Activities Found in Human Tears
Ophthalmology, 1981Human tears were found to inhibit the thiol-dependent protease, papain. Inhibitory activity in normal tears was compared with that in patients with blepharitis, infectious and allergic conjunctivitis, and herpes simplex. Activities lower than normal were found in some patients with infectious conjunctivitis and blepharitis.
J A, Anderson, I H, Leopold
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Antiproliferative effect and antiproteolytic activity of tetra-behzamidine derivatives
The Journal of Steroid Biochemistry, 1987Roberto Gambari, Paolo Ascenzi
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ANTIPROTEOLYTIC ACTIVITY OF SERUM FROM DOGS WITH EXPERIMENTALLY-INDUCED PEPTIC ULCERS
American Journal of Physiology, 1950E E, CLIFFTON, L E, YOUNG
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Proteolytic and antiproteolytic activities in goat antral follicles
Animal Reproduction Science, 1990Abstract Goat antral follicles were dissected and classified initially by size into three groups: 6 mm. Follicles less than 3 mm diameter were studied without any further classification. All others were classified according to their gross stereoscopic microscope appearance into four sub-groups.
A.M. Rosales +4 more
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Aromatic tetra-amidines: synthesis of halo-derivatives and their antiproteolytic activity.
Il Farmaco; edizione scientifica, 1984Mono-halo derivatives of 1,3-di-(p-amidinophenoxy)-2,2-bis-(p-amidinophenoxymethyl)p ropane (TAPP-H) have been synthesized and their inhibitory effect on the bovine trypsin, bovine thrombin and porcine pancreatic kallikrein catalyzed hydrolysis of p-nitroanilides of amino acids was investigated, at pH 8.1 and 37 degrees, in parallel with that of TAPP-H
FERRONI R +6 more
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