Results 181 to 190 of about 4,292 (206)

2-Benzazepines. 5. Synthesis of pyrimido[5,4-d][2]benzazepines and their evaluation as anxiolytic agents

Journal of Medicinal Chemistry, 1983
A series of 5H-pyrimido[5,4-d][2]benzazepines has been synthesized, starting from the corresponding 2-benzazepin-5-ones, and evaluated as potential anxiolytic agents. Selected compounds from this series show a pharmacological profile of action different than that of diazepam. They are more potent than diazepam in the anti-pentylenetetrazole test and in
J. Sepinwall, Earley Jv, Fryer Ri, Eugene John Trybulski, Reeder E, Armin Walser, W. D. Horst, Louis E. Benjamin, A. B. Davidson, Norman W. Gilman   +9 more
openaire   +3 more sources

ChemInform Abstract: 2‐Benzazepines. Part 9. Synthesis and Chemistry of 3H‐2‐Benzazepine and Pyrimido(4,5‐d)(2)benzazepine Derivatives.

ChemInform, 1987
AbstractThe benzazepines (II), prepared from the acetylenes (I), are transformed into the isomeric esters (VI) and (VII) by consecutive bromination, dehydrobromination, and palladium‐catalyzed alkoxycarbonylation.
L. Todaro, Eugene J. Trybulski, Rodney Ian Fryer, S. Vitone, Earl Reeder   +4 more
openaire   +2 more sources

Synthesis and Biological Evaluation of Benzazepine Oxazolidinone Antibacterials.

ChemInform, 2003
AbstractFor Abstract see ChemInform Abstract in Full Text.
Betty H. Yagi, Judith C. Hamel, Paul D. Johnson, Ford Charles W, Douglas Stapert, Gary E. Zurenko, Ronda D. Schaadt, Judy K. Moerman, Paul Adrian Aristoff   +8 more
openaire   +4 more sources

Synthesis of Spiro[benzazepine-2,4‘-piperidine]

The Journal of Organic Chemistry, 1998
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
D. Gomez Pardo, J.-L. Peglion and, Aimee Dessinges, Janine Cossy, C. Poitevin† and   +4 more
openaire   +3 more sources

Synthesis of a [2]benzazepine analogue of clavizepine

Tetrahedron Letters, 2001
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
Domingo Domínguez, Alberto Garcı́a, Sonia Paz   +2 more
openaire   +3 more sources

ChemInform Abstract: Novel Synthesis of the 2‐Benzazepine System

ChemInform, 1999
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
V. M. Kisel, E. O. Kostyrko, V. A. Kovtunenko   +2 more
openaire   +3 more sources

A free radical route to the benzazepines and dibenzazepines

Tetrahedron Letters, 1993
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
Zhizhen Barbara Zheng, Paul Dowd
openaire   +3 more sources

Synthesis and Properties of New Functionalized 2‐Benzazepines.

ChemInform, 2006
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
V. M. Kysil, V. A. Kovtunenko, E. O. Kostyrko   +2 more
openaire   +3 more sources

Regioselective alkylation reactions of 2,4-diphenyl-3H-1-benzazepine give either 3-alkyl-3H-1-benzazepines or 1-alkyl-1H-1-benzazepines

Tetrahedron Letters, 2014
AbstractDeprotonation of benzazepine (I) followed by reaction with alkyl halides or tosylates give either products of alkylation at C3 or at the nitrogen as well as mixtures of both types of products.
Allen Ko, Gopal Subramaniam, David J. Szalda, Aaron Lam, Jeffrey Li, Sasan Karimi, Edyta M. Greer, Keith Ramig   +7 more
openaire   +3 more sources

ChemInform Abstract: A Palladium‐Catalyzed Domino Process to 1‐Benzazepines. [PDF]

ChemInform, 1998
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
Gerald Dyker, Hardy Markwitz
openaire   +2 more sources