Results 121 to 130 of about 8,103 (214)

SYNTHESIS, CHARACTERIZATION AND ANTIMICROBIAL STUDY OF SOME BENZENESULFONAMIDE BASED BIPYRAZOLES

, 2014
Objectives: To synthesize, characterize and evaluate antimicrobial properties of some benzenesulfonamide based bipyrazole. Methods: The benzenesulfonamide based bipyrazole 1a-d & 2a-f have been synthesized by the reaction between 1-[1-aryl ...
Sharma, Pawan K., Singh, Karan
core  

Reaction of mesoionic compounds deriving from cyclic N-acyl-alpha-aminoacids with N-(phenylmethylene)benzenesulfonamide

, 1999
We studied the behaviour of bicyclic mesoionic compounds derived from the cyclodehydration of cyclic N-acyl-α-aminoacids 1-4 with N- (phenylmethylene)benzenesulfonamide 5. The reaction affords spirocyclic β- lactams and/or imidazo-condensed products (the
C. La Rosa, P. Dalla Croce, R. Ferraccioli   +2 more
core   +1 more source

Designing, synthesis and bioactivities of 4-[3-(4-hydroxyphenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]benzenesulfonamides

Journal of Enzyme Inhibition and Medicinal Chemistry, 2017
In this study, 4-[3-(4-hydroxyphenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]benzenesulfonamide (1–9) types compounds were synthesized and their chemical structures were confirmed by 1H NMR, 13C NMR and HRMS spectra.
Halise Inci Gul, Ebru Mete, Sakip Emre Eren, Hiroshi Sakagami, Cem Yamali, Claudiu T. Supuran   +5 more
doaj   +1 more source

Synthesis of Anti-Microtubule N-(2-Arylindol-7-yl)benzenesulfonamide Derivatives and Their Antitumor Mechanisms

, 2010
Breaking the cycle: A series of N-(2-arylindol-7-yl)benzenesulfonamide derivatives were prepared. Among them, compound 2 showed promising antiproliferative activity against hormone-resistant prostate cancer PC-3 cells, induced G2/M-phase arrest, and ...
Chen, Grace Shiahuy, Li, Huoming, Huoming Li, Chern, Ji Wang, Chun-Tang Chiou, Wei-Ming Dai, Chiou, Chun Tang, Grace Shiahuy Chen, Lei Shi, Chen, Meng Ling, Dai, Wei Ming, Xiang-Hong Huang, Meng-Ling Chen, Huang, Xiang Hong, Shi, Lei, Ji-Wang Chern   +15 more
core   +1 more source

Benzenesulfonamide

Acta Crystallographica Section E Structure Reports Online, 2007
B. Thimme Gowda, Roopa Nayak, Jozef Kožíšek, Miroslav Tokarčík, Hartmut Fuess   +4 more
openaire   +1 more source

Docking study of novel designed indazole derivatives against topoisomerase-II DNA gyrase enzyme for antibacterial screening

Intelligent Pharmacy
Aim of the study was designed for the design of novel indazole derivatives and evaluation of their docking against topoisomerase-II DNA gyrase enzyme for the antibacterial screening. Different novel substituted indazol-3-yl benzenesulfonamide derivatives
Nabeela Mareyam, Md Nematullah, Md Faheem Haider, Md Akbar, Md Azizur Rahman   +4 more
doaj   +1 more source

Synthesis, antimicrobial and QSAR studies of novel benzenesulfonamide derivatives [PDF]

, 2018
852-857Novel benzenesulfonamide derivatives have been synthesized and characterized by various spectroscopical and analytical techniques, such as, FT-IR, UV-Vis, and NMR, and elemental analysis.
Dığrak, Metin, Turkmen, Hasan, Zengin, Huseyin, Zengin, Gulay   +3 more
core  

(S)-(−)-4-[4-[2-(Isochroman-1-yl)ethyl]piperazin-1-yl]benzenesulfonamide, a Selective Dopamine D₄ Antagonist

, 2016
(S)-(−)-4-[4-[2-(Isochroman-1-yl)ethyl]piperazin-1-yl]benzenesulfonamide, a Selective Dopamine D4 ...
Robert A. Lahti (3018411), Martin W. Smith (2068087), Iain J. Martin (3018414), R. M. Huff (3018408), Charles F. Lawson (3018417), John C. Sih (3010380), Siusaidh K. Schlachter (3018402), Ruth E. TenBrink (3018399), Carol L. Bergh (3018423), J. Neil Duncan (3012621), Douglas W. Harris (3018420), Barry S. Lutzke (3018396), Susan A. Rees (3018405)   +12 more
core   +1 more source

An overlap of interacting amino acid in cluster I & II with inositol-(1,3,4,5)-tetrakisphosphate, benzenesulfonamide and sulfonamide derivatives within Akt2 binding cavity.

, 2016
An overlap of interacting amino acid in cluster I & II with inositol-(1,3,4,5)-tetrakisphosphate, benzenesulfonamide and sulfonamide derivatives within Akt2 binding cavity.
Noreen Akhtar (3609425), Ishrat Jabeen (1284885)   +1 more
core   +1 more source

The evaluation of pharmacokinetic parameters of 4-(5-methyl-1,3,4-oxadiazole-2-yl)- benzenesulfonamide and its metabolites in rat plasma

4-(5-methyl-1,3,4-oxadiazole-2-yl)-benzenesulfonamide (ODASA) is a new pharmacologically active compound, which is capable of reducing intraocular pressure by inhibiting carbonic anhydrase ...
Korsakov, M. K., Volkhin, N. N., Shetnev, A. A., Yaichkov, I. I., Khokhlov, A. L.   +4 more
core   +1 more source