Results 1 to 10 of about 59,564 (376)

2,2-difluorovinyl benzoates for diverse synthesis of gem-difluoroenol ethers by Ni-catalyzed cross-coupling reactions

open access: yesNature Communications, 2021
The gem-difluoroalkene functionality is relevant to drug design as it is a bioisostere of a carbonyl group. Here, the authors report the synthesis of 2,2-difluorovinyl benzoates as versatile building blocks for modular synthesis of gem-difluoroenol ...
Bingnan Du   +6 more
doaj   +2 more sources

Glycosyl ortho-(1-phenylvinyl)benzoates versatile glycosyl donors for highly efficient synthesis of both O-glycosides and nucleosides

open access: yesNature Communications, 2020
O-glycosides and nucleosides are important biomolecules. Here, the authors developed a protocol for the synthesis of such molecules with a broad substrate scope using glycosyl ortho-(1-phenylvinyl)benzoates as glycosyl donors that allow for mild reaction
Penghua Li   +8 more
doaj   +2 more sources

Low-Valent Tungsten Catalyzed Carbonylative Synthesis of Benzoates from Aryl Iodides and Alcohols [PDF]

open access: yesMolecules
Non-noble metals catalyzed carbonylative reactions serve as straightforward and sustainable methods for the synthesis of functionalized carbonyl-containing compounds.
Feihua Ye   +6 more
doaj   +2 more sources

Comparative Antibacterial Activities of Some Monosaccharide and Disaccharide Benzoates

open access: yesOrbital: The Electronic Journal of Chemistry, 2015
For comparative antibacterial studies a number of furanose (3, 5), pyranose (7, 9, 11, 13), and disaccharide benzoates (14, 15) were prepared by direct benzoylation method.
Mohammed M. Matin   +3 more
doaj   +4 more sources

Antibacterial Activity of Salicylanilide 4-(Trifluoromethyl)-benzoates

open access: yesMolecules, 2013
The development of novel antimicrobial agents represents a timely research topic. Eighteen salicylanilide 4-(trifluoromethyl)benzoates were evaluated against Mycobacterium tuberculosis, M. avium and M.
Jiřina Stolaříková   +5 more
doaj   +2 more sources

Antimycobacterial Assessment of Salicylanilide Benzoates including Multidrug-Resistant Tuberculosis Strains

open access: yesMolecules, 2012
The increasing emergence especially of drug-resistant tuberculosis has led to a strong demand for new anti-tuberculosis drugs. Eighteen salicylanilide benzoates were evaluated for their inhibition potential against Mycobacterium tuberculosis ...
Jiřina Stolaříková   +2 more
doaj   +2 more sources

Enantioselective synthesis of γ-chiral amides via copper-catalyzed reductive relay hydroaminocarbonylation [PDF]

open access: yesNature Communications
Chiral amides are common and effective structural motifs found in many pharmaceuticals and biologically active molecules. Despite their importance, existing synthetic methods are predominantly employed for the synthesis of α-amides and β-amides.
Yang Yuan, Youcan Zhang, Xiao-Feng Wu
doaj   +2 more sources

In Vitro Antibacterial and Antifungal Activity of Salicylanilide Benzoates

open access: yesThe Scientific World Journal, 2012
The resistance to antimicrobial agents brings a need of novel antimicrobial agents. We have synthesized and found the in vitro antibacterial activity of salicylanilide esters with benzoic acid (2-(phenylcarbamoyl)phenyl benzoates) in micromolar range ...
Martin Krátký   +2 more
doaj   +2 more sources

Floral scent components in Rhododendron fortunei and its regulation by gene expression of S-adenosyl-l-methionine: benzoic acid carboxyl methyl transferase (BAMT) [PDF]

open access: yesCiência Rural, 2023
: Rhododendron fortune belongs to a scented Rhododendron species native to China, which produces fragrant flowers of great ornamental and environmental values for landscaping or indoor beautification.
Chen FeiZhang   +9 more
doaj   +1 more source

Nitrobenzoates and Nitrothiobenzoates with Activity against M. tuberculosis

open access: yesMicroorganisms, 2023
Esters of weak acids have shown improved antimycobacterial activity over the corresponding free acids and nitro benzoates in particular have previously shown to have a very intriguing activity. To expand the potential of nitro-derivatives of benzoic acid
João P. Pais   +6 more
doaj   +1 more source

Home - About - Disclaimer - Privacy