Results 1 to 10 of about 59,564 (376)
The gem-difluoroalkene functionality is relevant to drug design as it is a bioisostere of a carbonyl group. Here, the authors report the synthesis of 2,2-difluorovinyl benzoates as versatile building blocks for modular synthesis of gem-difluoroenol ...
Bingnan Du+6 more
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O-glycosides and nucleosides are important biomolecules. Here, the authors developed a protocol for the synthesis of such molecules with a broad substrate scope using glycosyl ortho-(1-phenylvinyl)benzoates as glycosyl donors that allow for mild reaction
Penghua Li+8 more
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Low-Valent Tungsten Catalyzed Carbonylative Synthesis of Benzoates from Aryl Iodides and Alcohols [PDF]
Non-noble metals catalyzed carbonylative reactions serve as straightforward and sustainable methods for the synthesis of functionalized carbonyl-containing compounds.
Feihua Ye+6 more
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Comparative Antibacterial Activities of Some Monosaccharide and Disaccharide Benzoates
For comparative antibacterial studies a number of furanose (3, 5), pyranose (7, 9, 11, 13), and disaccharide benzoates (14, 15) were prepared by direct benzoylation method.
Mohammed M. Matin+3 more
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Antibacterial Activity of Salicylanilide 4-(Trifluoromethyl)-benzoates
The development of novel antimicrobial agents represents a timely research topic. Eighteen salicylanilide 4-(trifluoromethyl)benzoates were evaluated against Mycobacterium tuberculosis, M. avium and M.
Jiřina Stolaříková+5 more
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The increasing emergence especially of drug-resistant tuberculosis has led to a strong demand for new anti-tuberculosis drugs. Eighteen salicylanilide benzoates were evaluated for their inhibition potential against Mycobacterium tuberculosis ...
Jiřina Stolaříková+2 more
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Enantioselective synthesis of γ-chiral amides via copper-catalyzed reductive relay hydroaminocarbonylation [PDF]
Chiral amides are common and effective structural motifs found in many pharmaceuticals and biologically active molecules. Despite their importance, existing synthetic methods are predominantly employed for the synthesis of α-amides and β-amides.
Yang Yuan, Youcan Zhang, Xiao-Feng Wu
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In Vitro Antibacterial and Antifungal Activity of Salicylanilide Benzoates
The resistance to antimicrobial agents brings a need of novel antimicrobial agents. We have synthesized and found the in vitro antibacterial activity of salicylanilide esters with benzoic acid (2-(phenylcarbamoyl)phenyl benzoates) in micromolar range ...
Martin Krátký+2 more
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Floral scent components in Rhododendron fortunei and its regulation by gene expression of S-adenosyl-l-methionine: benzoic acid carboxyl methyl transferase (BAMT) [PDF]
: Rhododendron fortune belongs to a scented Rhododendron species native to China, which produces fragrant flowers of great ornamental and environmental values for landscaping or indoor beautification.
Chen FeiZhang+9 more
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Nitrobenzoates and Nitrothiobenzoates with Activity against M. tuberculosis
Esters of weak acids have shown improved antimycobacterial activity over the corresponding free acids and nitro benzoates in particular have previously shown to have a very intriguing activity. To expand the potential of nitro-derivatives of benzoic acid
João P. Pais+6 more
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