Results 101 to 110 of about 10,895 (224)

SYNTHESIS AND CHEMICAL CHARACTERIZATION OF BENZIMIDAZOLE FUSED BENZOPYRAN DERIVATIVES AND EVALUATION OF THEIR ANTI-BACTERIAL POTENCY

, 2019
Benz-imidazole fused benzopyran derivatives were prepared by the reaction of 2-(1H-Benzo[d]Imidazol-2-yl)-1phenyl-1H-Benzo[f]chromeno-3-amine with different substituted benzaldehydes.
Rufaida Farheen *, Y. Rajesh Babu 1
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Cis-glyco-fused benzopyran derivatives as hit compounds for the development of therapeutic and diagnostic tools against neurodegenerative diseases

, 2014
Oligomeric and fibrillar aggregates generated by amyloid-β (Aβ) and prion protein (PrP) peptides are amongst the principal components of amyloid plaques found post mortem in patients suffering from Alzheimer's disease and mammalian prion diseases.
Sironi E., Martorana A. M., Airoldi C., Merlo S., Cardona F., Salmona M., Colombo L., La Ferla B.   +7 more
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3-Hemiacetals of 3,4-Dihydrospiro[2H-1-benzopyran-2,1'(3'H)-isobenzofuran]-3,4-dione

, 1975
Oxidation of 2?-hydroxymethylfiavonol with periodic acid in methanol gives 3,4-dihydro-3-hydroxy-3-methoxyspiro[2H-1-benzopyran-2,1'(3'H)- isobenzofuran]-4-one.
EJ McGarry, JW Clark-Lewis
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Synthesis of Deuterated Benzopyran Derivatives as Selective COX‑2 Inhibitors with Improved Pharmacokinetic Properties

, 2016
We designed a series of specifically deuterated benzopyran analogues as new COX-2 inhibitors with the aim of improving their pharmacokinetic properties. As expected, the deuterated compounds retained potency and selectivity for COX-2.
Jianqi Liu (1738939), Micky D. Tortorella (1515469), Yang Bai (198601), Yican Wang (1738942), Zhengchao Tu (542105), John J. Talley (1515478), Xiaorong Liu (239247), Dingsheng Wen (1738933), Yanmei Zhang (122913), Yongzhi Lu (1738936), Xin Lu (24821)   +10 more
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In-Silico Study, Synthesis and Pharmacological Screening of Novel Benzopyran-3-Carbonyl Derivatives as Antidiabetic Agents

Introduction: In the current work, in-silico docking investigation for 60 benzopyran-3-carbonyl derivatives was conducted since benzopyran derivatives play a vital role in many different research disciplines.
Bhartendu Sharma, Ranjit Singh
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Synthesis of Some New Heteroarylamino-3-Nitro-2H-[1]-Benzopyran-2-ones and their Antibacterial Activity

, 2016
Novel derivatives of benzopyran-2-ones are synthesized by catalytic condensation reaction. 4-(3-Hydroxy-2-pyridinylamino)- 3-nitro-2H-[1]-benzopyran-2-one  4a,  4-(4-methyl-3-nitro-2-pyridinylamino)-3-nitro-2H-[1]-benzopyran-2-one,  4b  and 4 ...
Ismaili, Hamit, Thaci, Veprim, Vehapi, Idriz, Hoti, Ramiz, Mulliqi-Osmani, Gjyle   +4 more
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Modulation of Vascular Reactivity by Novel Synthetic Benzopyran Analogues in Rat Aortas

, 2016
A substantial body of research described ATP-dependent potassium (K ATP ) channels, sarcolemmal and mitochondrial, with different physiological functions and pharmacological behaviour in various tissues (pancreatic â-cells, brain, skeletal muscle and
Bedreag, O., Petrus, A., Duicu, O., Jost, Norbert László, Baczkó, István, Kiss, Loránd, Sturza, A., Utu, D.   +7 more
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Neuropharmacological Profile of Novel Benzopyran-2-One Derivatives in Experimental Mice

, 2019
The present study was aimed to assess the neuropharmacological properties of the novel Benzopyran-2-one (coumarin) derivatives i.e., 7-(2-(m-nitro)-phenyl thiazolidinyl)-4-methyl benzopyran-2-one (comp-I), 7-(2-(o,p-dichloro)-phenyl thiazolidinyl)-4 ...
Kumar, Umesh
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Synthesis and antimicrobial screening of 2,4-diaryl-6-[2' H-[1']-4'-hydroxy-2'-oxo benzopyran-3'-yl]pyridines and 2,6-diaryl-4-[2' H-[1']-4' -hydroxy-2' -oxo-benzopyran-3'yl]pyridines

, 2004
2727-2730The chalcones of 4-hydroxycoumarin such as 4-hydroxy-2-oxo-3-(1'-oxo-3'-phenylprop-2'-enyl)-2H-[1]-benzopyran 1 and 4-hydroxy-2-oxo-3-(3'-oxo-3'-phenylprop-1'-enyl)-2H-[1]-benzopyran 2 are separately refluxed with phenacyl pyridinium bromide ...
Mulwad, V V, Satwe, D S
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Studies in Hantrsch thiazole synthesis:Synthesis of 3-(2-allylamino-4-thiazolyl)-2H-1- benzopyran-2-ones and 3-(4-phenylthiazoline-2-anil)-2H-1-benzopyran-2-ones in solid state

, 2003
1738-1741Interaction of 3-(2-bromoacetyl)coumarins with N-allylthiourea and diphenyl thiourea in solid state furnish corresponding 3-(2-allyl amino-4-thiazolyl)-2H-1-benzopyran-2-ones and 3-(4-phenyl thiazoline-2-anil )-2H-1-benzopyran-2-ones.
Rao, V Rajeswar, Reddy, R Vinod, Kumar, P Vijay   +2 more
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