Results 21 to 30 of about 6,109 (244)
Antimicrobial Potential of Carbazole Derivatives
Croatica Chemica Acta, 2022 Amongst many nitrogen-containing heterocycles, carbazole frame is the building block of various biologically active compounds, including both synthetic and natural products of which its antimicrobial and antifungal activities are the most examined. In this review, 3, 4 and N- substituted carbazole derivatives and their antimicrobial activities are ...
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Synthesis, characterization and biological evaluation of some newer carbazole derivatives [PDF]
Journal of the Serbian Chemical Society, 2014 A series of novel 5-((9H-carbazol-9-yl)methyl)-N-((substituted phenyl)(piperazin-1-yl)methyl)-1,3,4-oxadiazol-2-amine (4a-4o) derivatives was synthesized by starting with carbazole which on reaction with ethyl choloroacetate yielded ethyl 2-(9H ...
Sharma Divyanshu +2 more
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Sulfonamido-derivatives of unsubstituted carbazoles as BACE1 inhibitors [PDF]
Bioorganic & Medicinal Chemistry Letters, 2017 A novel series of variously substituted N-[3-(9H-carbazol-9-yl)-2-hydroxypropyl]-arylsulfonamides has been synthesized and assayed for β-Secretase (BACE1) inhibitory activity. BACE1 is a widely recognized drug target for the prevention and treatment of Alzheimer's Disease (AD).
BERTINI, SIMONE +11 more
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Facile synthesis of indolo[3,2-a]carbazoles via Pd-catalyzed twofold oxidative cyclization
Beilstein Journal of Organic Chemistry, 2016 A rapid and efficient route has been developed for the synthesis of 9-methoxycarbonylindolo[3,2-a]carbazole derivatives. The key steps in this approach involved an aromatic amination and an oxidative biaryl coupling.
Chao Yang +4 more
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LXXIII.—N-Acyl derivatives of carbazole [PDF]
J. Chem. Soc., Trans., 1918 n ...
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Carbazole scaffolds in cancer therapy: a review from 2012 to 2018
Journal of Enzyme Inhibition and Medicinal Chemistry, 2019 For over half a century, the carbazole skeleton has been the key structural motif of many biologically active compounds including natural and synthetic products.
Samar Issa +6 more
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Frontiers in Chemistry, 2019 Difluoroboron-dipyrromethenes (BODIPYs) are highly popular fluorescent dyes with applications as NIR probes for bioimaging, fluorescent tags/sensors and as photosensitizers in cancer therapy and organic photovoltaics.
Iti Gupta, Praseetha E. Kesavan
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Разработка и регистрация лекарственных средств, 2020 Introduction. Currently, more than 600 thousand people a year are affected by malignant tumors on the territory of the Russian Federation. Despite the large selection of antitumor drugs and the variety of mechanisms of their action, the effectiveness of ...
D. A. Kozin +5 more
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Synthesis of oxadiazole substituted new carbazole derivatives as antioxidant and antiurease agent
European Journal of Biological Research, 2022 Heterocyclic compounds containing nitrogen together with an oxygen atom in their structures are an important class of medicinal chemistry compounds due to their interesting diverse biological applications.
Nurhan Gümrükçüoğlu +1 more
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MoleculesCarbazole-based molecules play a significant role in dye-sensitized solar cells (DSSCs) due to their advantageous properties. Carbazole derivatives are known for their thermal stability, high hole-transport capability, electron-rich (p-type ...
Ayagoz Ibrayeva +5 more
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