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ChemMedChem, Volume 21, Issue 16, 27 August 2026.We explore covalent allosteric targeting of MGL regulatory cysteines using iso‐ and benzisothiazolinone scaffolds. Combining mechanism‐based warhead release with structure‐guided scaffold decoration to improve molecular recognition, this study probes strategies to achieve selective on‐target engagement beyond the catalytic site. Monoacylglycerol lipase
Edoardo Rocca +12 more
wiley +1 more source
Agonist D2-dopamine receptors reduces hemoconcentration in hyperstimulated women undergoing assisted reproduction [PDF]
Гинекология, 2014 Background. Ovarian hyperstimulation syndrome (OHSS) results from increased vascular permeability (VP) caused by ovarian hypersecretion of vascular endothelial growth factor (VEGF), which activates its receptor-2.
S V Fetisova, I E Korneeva, T U Ivaniec
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Journal of Pain Research, 2018 Xiao-Cui Yuan,1 Qiang Wang,2 Wen Su,3 Hong-Ping Li,1 Cai-Hua Wu,3 Fang Gao,1 Hong-Chun Xiang,1 He Zhu,1 Li-Xue Lin,1 Xue-Fei Hu,1 Jie Cao,4 Jing-Jing Li,1 Man Li1 1Department of Neurobiology and Key Laboratory of Neurological Diseases of Ministry of ...
Yuan X +12 more
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Cannabinoid CB1 receptor; cannabinoid CB2 receptor [PDF]
Science-Business eXchange, 2008 openaire +1 more source
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Arylsulfonamide CB2 receptor agonists: SAR and optimization of CB2 selectivity
Bioorganic and Medicinal Chemistry Letters, 2008A high-throughput screening campaign resulted in the discovery of a highly potent dual cannabinoid receptor 1 (CB1) and 2 (CB2) agonist. Following a thorough SAR exploration, a series of selective CB2 full agonists were identified.
Brian Dymock +2 more
exaly +3 more sources