Results 161 to 170 of about 19,626 (172)

Design, synthesis and biological evaluation of novel DNA gyrase inhibitors and their siderophore mimic conjugates

Bioorganic Chemistry, 2020
ANDRAŽ Lamut, Cristina D Cruz, Ziga Skok   +2 more
exaly  

Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitors

Bioorganic and Medicinal Chemistry, 2017
Tihomir Tomasic, Michaela Barančoková, Janez Ilas   +2 more
exaly  

Synthesis and Evaluation of N‐Phenylpyrrolamides as DNA Gyrase B Inhibitors

ChemMedChem, 2018
Martina Ďurčík, Päivi Tammela, Michaela Barančoková   +2 more
exaly  

In silico fragment-based discovery of indolin-2-one analogues as potent DNA gyrase inhibitors

Bioorganic and Medicinal Chemistry Letters, 2005
Simona Golic Grdadolnik, Roman Jerala, Metka Filipic   +2 more
exaly  

DNA Gyrase Is the Target for the Quinolone Drug Ciprofloxacin in Arabidopsis thaliana

Journal of Biological Chemistry, 2016
Lesley A Mitchenall, Joshua S Mylne, Anthony Maxwell   +2 more
exaly  

DNA-induced narrowing of the gyrase N-gate coordinates T-segment capture and strand passage

Proceedings of the National Academy of Sciences of the United States of America, 2011
Airat Gubaev, Dagmar Klostermeier, Klostermeier Dagmar   +2 more
exaly  

DNA gyrase and the mechanism of DNA supercoiling

Biochemical Society Transactions, 1999
openaire   +1 more source

Fragment-based discovery of DNA gyrase inhibitors targeting the ATPase subunit of GyrB

Bioorganic and Medicinal Chemistry Letters, 2016
Michael F Mesleh, Jason B Cross, Terence I Moy   +2 more
exaly  

Thirty years of Escherichia coli DNA gyrase: From in vivo function to single-molecule mechanism

Biochimie, 2007
Marcelo Nollmann, Nancy J Crisona, Paola B Arimondo   +2 more
exaly  

New N -phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity

European Journal of Medicinal Chemistry, 2018
Martina Ďurčík, Denise Lovison, Ziga Skok   +2 more
exaly