Results 11 to 20 of about 12,682 (158)
Tropical and Subtropical Agroecosystems, 2023 Background: During the last few years the home box transcription factor WUSCHEL (WUS) has been shown to cause dedifferentiation when expressed on somatic cells followed by a production of new stem cells that can lead to somatic embryogenesis or ...
Ana Ly Arroyo Herrera +7 more
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Molecules, 2022 Hybridization of steroids and other pharmacophores often modifies the bioactivity of the parent compounds, improving selectivity and side effect profile.
Ferenc Kovács +5 more
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Retention behaviour of some estradiol derivatives on alumina in normal phase chromatrography [PDF]
Journal of the Serbian Chemical Society, 2003 The retention constants of variously substituted estradiol derivatives were measured as a function of the composition of various binary mobile phases in order to study the relationship between chemical structure and retention behavior in TLC on alumina ...
Ačanski Marijana M.
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Holographic QSAR of estradiol derivatives
Science Bulletin, 2003 Holographic QSAR model is constructed to predict relative binding affinities of estradiol derivatives with lamb uterine estrogen receptor. The method does not require the generation of three-dimensional structure of the compounds. The factors that influence the quality of QSAR model are discussed.
Shihai Cui +3 more
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Chemometric estimation of the retention behavior of selected estradiol derivatives [PDF]
Acta Periodica Technologica, 2015 Quantitative structure-retention relationship (QSRR) analysis has been performed in order to correlate the retention of selected estradiol derivatives with their calculated molecular lipophilicity.
Karadžić Milica Ž. +5 more
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Frontiers in Molecular Biosciences, 2021 The treatment of common steroids: estrone, estradiol, cortisol, and pregnenolone with tributylsulfoammonium betaine (TBSAB) provides a convenient chemoselective conversion of the steroids alcohol/phenol moiety to the corresponding steroidal organosulfate.
Jaber A. Alshehri +2 more
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Molecules, 2010 Combinatorial chemistry is a powerful tool used to rapidly generate a large number of potentially biologically active compounds. In our goal to develop bisubstrate inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) that interact with both ...
Donald Poirier +2 more
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Estradiol regulation of nucleotidases in female reproductive tract epithelial cells and fibroblasts. [PDF]
PLoS ONE, 2013 The use of topical and oral adenosine derivatives in HIV prevention that need to be maintained in tissues and cells at effective levels to prevent transmission prompted us to ask whether estradiol could influence the regulation of catabolic nucleotidase ...
Zheng Shen +7 more
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Applied Sciences, 2022 C-Ring oxidized estrone acetate derivatives as antiproliferative agents were prepared and tested against five cancer cell lines by the 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide assay.
Catarina Canário +7 more
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Targeting the estrogen receptor with metal-carbonyl derivatives of estradiol [PDF]
Bioorganic & Medicinal Chemistry Letters, 2012 As part of our program to develop new probes for the estrogen receptor binding domain, we prepared and evaluated a novel 17α-(rhenium tricarbonyl bipyridyl) vinyl estradiol complex. Preparation of the final compound was achieved using the Stille coupling between the preformed brominated rhenium tricarbonyl bipyridine complex and the tributylstannyl ...
Robert N, Hanson +7 more
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