Results 111 to 120 of about 5,945,207 (220)

The effects of serum, lithium, ethacrynic acid, and a low external concentration of potassium on specific [3H]-ouabain binding to human lymphocytes after incubation for 3 days.

, 1986
We have quantified specific [3H]-ouabain binding sites in normal human lymphocytes, and have measured the changes in the numbers of those sites which occur in response to various stimuli.
Harper, C, Aronson, JK, Aronson, Jeffrey, Grahame-Smith, DG, Rapeport, WG   +4 more
core   +1 more source

Arene Ruthenium Complexes with Ethacrynic Acid-Modified Ligands: Synthesis, Characterization and Antiproliferative Activity

, 2016
Ethacrynic acid is a broad acting glutathione transferase inhibitor, and its incorporation within suitable metal complexes results in enhancement of the anticancer activity.1 A series of pyridine- and phosphine-based ligands functionalized with ...
Biancalana, L., Zacchini, S., ZACCHINI, STEFANO, Chiellini, F., Dyson, P. J., Gabbiani, C., AGONIGI, GABRIELE, GABBIANI, CHIARA, Dyson, Paul J., PAMPALONI, GUIDO, Pampaloni, G., CHIELLINI, FEDERICA, Riedel, T., Marchetti, F., Agonigi, G., FUNAIOLI, TIZIANA, MARCHETTI, FABIO, BIANCALANA, LORENZO, Funaioli, T.   +18 more
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Influence of Ethacrynic Acid on Muscle Surface Enzymes and of Ethacrynic Acid and Ouabain on Na, K, and H₂O in Frog Muscle

, 1972
Isolated frog muscles were exposed to concentrations of ethacrynic acid (2,3-dichloro-4-(2-methylene-butyryl)phenoxyaceticacid)ranging from 10−8 to 10−2 M.
T. S. Still, J. R. Riordan, J. F. Manery, E. E. Dryden   +3 more
core   +1 more source

Synthesis and Cytotoxic Activity of Ruthenium Complexes with Ethacrynic Acid Derived Ligands

, 2015
There is currently high interest in the design of organic motifs containing biologically-active fragments to be incorporated within suitable metal complexes, in order to confer them enhanced anticancer activity. One of the possible approaches regards the
Biancalana, L., Zacchini, S., ZACCHINI, STEFANO, Dyson, P. J., Dyson, Paul J., Agonigi, Gabriele, PAMPALONI, GUIDO, Pampaloni, G., Riedel, T., Marchetti, F., Agonigi, G., Paunescu, E., MARCHETTI, FABIO, BIANCALANA, LORENZO   +13 more
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Effects of trifluoperazine, ouabain, and ethacrynic acid on intestinal calcium transport

, 1983
Bidirectional steady-state calcium fluxes were measured in vitro under short-circuited conditions in segments of rat duodenum and descending colon. The calcium-activated ATPase (Ca-ATPase) inhibitor trifluoperazine (TFP, 0.1 mM) reduced net calcium ...
E. Angeid-Backman, F. L. Coe, M. J. Favus, M. D. Breyer   +3 more
core   +1 more source

Inhibition of glutathione S-transferase activity in human melanoma cells by alfa, beta-unsaturated carbonyl derivatives : effects of acrolein, cinnamaldehyde, citral, crotonaldehyde, curcumin, ethacrynic acid, and trans-2-hexenal

, 1996
The glutathione S-transferase (GST) activity towards 1-chloro-2,4-dinitrobenzene in intact human IGR-39 melanoma cells was determined by the quantification by HPLC-analysis of the excreted glutathione (GSH) conjugate (S-(2,4-dinitrophenyl)glutathione ...
Bladeren, P.J. van, Amersfoort, C. van, Struik, I., Schefferlie, J.G., Ploemen, J.P.H.T.M., Keyzer, A.E., Iersel, M.L.P.S. van   +6 more
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Ruthenium arene complexes with triphenylphosphane ligands: cytotoxicity towards pancreatic cancer cells, interaction with model proteins, and effect of ethacrynic acid substitution

, 2017
L. Biancalana, A. Pratesi, F. Chiellini, S. Zacchini, T. Funaioli, C. Gabbiani, F. Marchetti   +6 more
semanticscholar   +1 more source

Synthesis and Antiproliferative Activity of New Ruthenium Complexes with Ethacrynic Acid-Modified Ligands

, 2016
Pyridine- and phosphine-based ligands modified with ethacrynic acid (EA, i.e. a broad acting glutathione transferase inhibitor) were prepared and coordinated to ruthenium(II)-arene complexes.1 All the compounds (ligands and complexes) were fully ...
Biancalana, L., Zacchini, S., ZACCHINI, STEFANO, Chiellini, F., Dyson, P. J., Gabbiani, C., AGONIGI, GABRIELE, GABBIANI, CHIARA, Dyson, Paul J., PAMPALONI, GUIDO, Pampaloni, G., CHIELLINI, FEDERICA, Riedel, T., Marchetti, F., Agonigi, G., FUNAIOLI, TIZIANA, MARCHETTI, FABIO, BIANCALANA, LORENZO, Funaioli, T.   +18 more
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[Ethacrynic acid]. [PDF]

Schweizerische medizinische Wochenschrift, 1968
openaire   +3 more sources

Bromocriptine-associated ototoxicity

, 1984
Three patients treated with bromocriptine for chronic hepatic encephalopathy showed audiometric evidence of bilateral sensori-neural hearing-loss. Audiometrically, the hearing improved in all three patients when the bromocriptine dosage was reduced, thus
Morgan, MY, Ballantyne, J, Lanthier, PL
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