Results 111 to 120 of about 5,882,080 (212)

Arrestin‐dependent but G‐protein coupled receptor kinase‐independent uncoupling of D2‐dopamine receptors [PDF]

, 2013
Jeremy Celver, Meenakshi Sharma, Vaidehi Thanawala, J. Christopher Octeau, Abraham Kovoor   +4 more
openalex   +1 more source

Systematic assessment of chemokine ligand bias at the human chemokine receptor CXCR2 indicates G protein bias over β-arrestin recruitment and receptor internalization

Cell Communication and Signaling
Background The human CXC chemokine receptor 2 (CXCR2) is a G protein-coupled receptor (GPCR) interacting with multiple chemokines (i.e., CXC chemokine ligands CXCL1-3 and CXCL5-8). It is involved in inflammatory diseases as well as cancer.
Katrijn Boon, Nathan Vanalken, Martyna Szpakowska, Andy Chevigné, Dominique Schols, Tom Van Loy   +5 more
doaj   +1 more source

Activation of ryanodine-sensitive calcium store drives pseudo-allergic dermatitis via Mas-related G protein-coupled receptor X2 in mast cells

, 2023
Zhao Wang, Xi Zhao, Hongmei Zhou, Delu Che, Xiaojie Du, Dan Ye, Weihui Zeng, Songmei Geng   +7 more
openalex   +1 more source

Subnanomolar MAS-related G protein-coupled receptor-X2/B2 antagonists with efficacy in human mast cells and disease models [PDF]

Ghazl Al Hamwi, Mohamad Wessam Alnouri, Sven Verdonck, Piotr Leonczak, Shaswati Chaki, Stefan Frischbutter, Pavel Kolkhir, Michaela Matthey, Christina Kopp, Marek Bednarski, Yvonne K. Riedel, Daniel Marx, Sophie Clemens, Vigneshwaran Namasivayam, Susanne Gattner, Dominik Thimm, Katharina Sylvester, Katharina Wolf, Andreas E. Kremer, Steven De Jonghe, Daniela Wenzel, Magdalena Kotańska, Hydar Ali, Piet Herdewijn, Christa E. Müller   +24 more
openalex   +1 more source

The Allosteric Mechanism of G-Protein-Coupled Receptors is Induced Fit, Not Conformational Selection. [PDF]

Bioessays
Asadollahi K, Gooley PR, Weikl TR.
europepmc   +1 more source

Stoichiometry of G protein subunits affects the Saccharomyces cerevisiae mating pheromone signal transduction pathway.

, 1990
Gary M. Cole, David E. Stone, S I Reed
openalex   +2 more sources

Single Nucleotide Polymorphisms in the G-Protein Coupled Receptor Kinase 5 (GRK5) Gene are associated with Plasma LDL-Cholesterol Levels in Humans [PDF]

, 2018
Stefan Lutz, Mathias Falcenberg, Fausto Machicao, Andreas Peter, Martin Kächele, Elko Randrianarisoa, Angela Lehn‐Stefan, Róbert Wágner, Jürgen Machann, Fritz Schick, Martin Heni, Axel Ullrich, Andreas Fritsche, Norbert Stefan, Hans‐Ulrich Häring, Harald Staiger, Kοnstantinos Kantartzis   +16 more
openalex   +1 more source

Purification and characterization of predominant G-protein from bovine lung membranes. Biochemical and immunochemical comparison with Gi1 and Go purified from brain [PDF]

, 1989
Yasunori Kanaho, Stanley T. Crooke, Jeffrey M. Stadel   +2 more
openalex   +1 more source

G protein-coupled receptor digital twins for precision and personalized medicine. [PDF]

Comput Struct Biotechnol J
Boeringer T, Pardo M, Craig CJ, Maudsley S.   +3 more
europepmc   +1 more source

Serum Activity Against G Protein–Coupled Receptors and Severity of Orthostatic Symptoms in Postural Orthostatic Tachycardia Syndrome [PDF]

, 2020
Isabella Kharraziha, Jonas Axelsson, Fabrizio Ricci, Giuseppe Di Martino, Margaretha Persson, Richard Sutton, Artur Fedorowski, Viktor Hamrefors   +7 more
openalex   +1 more source