Results 141 to 150 of about 35,308 (311)

Recent Results from the H1 Collaboration [PDF]

open access: yesarXiv, 2009
An overview of recent physics results from the H1 collaboration is given. The covered areas are: rare processes and searches for new physics, structure functions and inclusive measurements, heavy flavour production, QCD and hadronic final states, diffractive scattering.
arxiv  

Stimulation of Histamine H1 Receptor Up-Regulates Histamine H1 Receptor Itself Through Activation of Receptor Gene Transcription

open access: yesJournal of Pharmacological Sciences, 2007
Histamine is a major mediator in allergy acting mainly through the histamine H1 receptor (H1R). Although H1R up-regulation has been suggested as an important step for induction of allergic symptoms, little is known about the regulation of H1R level. Here
Asish K. Das   +10 more
doaj  

Pharmacology of Antihistamines

open access: yesWorld Allergy Organization Journal, 2011
This article reviews the molecular biology of the interaction of histamine with its H1-receptor and describes the concept that H1-antihistamines are not receptor antagonists but are inverse agonists i.e.
Diana S Church, MD, Martin K Church, PhD
doaj  

Effects of loratadine, a histamine H1 receptor antagonist, on the skeletal system of young male rats

open access: yesDrug Design, Development and Therapy, 2019
Joanna Folwarczna, Natalia Konarek, Karolina Freier, Dawid Karbowniczek, Piotr Londzin, Aleksandra Janas Department of Pharmacology, School of Pharmacy with the Division of Laboratory Medicine in Sosnowiec, Medical University of Silesia, Katowice ...
Folwarczna J   +5 more
doaj  

Influence of Epinastine Hydrochloride, an H1-Receptor Antagonist, on the Function of Mite Allergen-Pulsed Murine Bone Marrow-Derived Dendritic Cells In Vitro and In Vivo

open access: yesMediators of Inflammation, 2009
There is established concept that dendritic cells (DCs) play essential roles in the development of allergic immune responses. However, the influence of H1 receptor antagonists on DC functions is not well defined.
Ken-Zaburo Oshima   +4 more
doaj   +1 more source

The effect of polymorphic genetic markers CYP2С19(rs4244285and rs4986893), CYP2D6(rs3892097), ABCB1(rs1045642) on sedation during treatment with histamine H1-receptor antagonist [PDF]

open access: gold, 2020
V.B. Grishina   +5 more
openalex   +1 more source

Antagonistic AI [PDF]

open access: yesarXiv
The vast majority of discourse around AI development assumes that subservient, "moral" models aligned with "human values" are universally beneficial -- in short, that good AI is sycophantic AI. We explore the shadow of the sycophantic paradigm, a design space we term antagonistic AI: AI systems that are disagreeable, rude, interrupting, confrontational,
arxiv  

Histamine H1 receptor occupancy in human brains after single oral doses of histamine H1 antagonists measured by positron emission tomography

open access: yesBritish Journal of Pharmacology, 1995
K. Yanai   +7 more
semanticscholar   +1 more source

Anticonvulsant and procognitive properties of Novel Histamine H3 Receptor Antagonists in male adult rats [PDF]

open access: yes, 2016
To determine the potential of histamine H3 receptor (H3R) ligands as new antiepileptic and procognitive drugs, aromatic ether derivatives (1-12) belonging to the nonimidazole class of ligands, with high in-vitro binding affinity at human H3R, were tested
Saad, Ali Kassem
core   +1 more source

Compound 48/80, a histamine-depleting agent, blocks the protective effect of morphine against electroconvulsive shock in mice

open access: yesBrazilian Journal of Medical and Biological Research, 2000
We have shown that morphine has an anticonvulsive effect against maximal electroconvulsive shock (MES) in mice, and this effect is antagonized by histamine H1-receptor antagonists.
Karadag C.H.   +4 more
doaj  

Home - About - Disclaimer - Privacy