Results 181 to 190 of about 42,534 (266)

Carbamoyl Pyridone HIV-1 Integrase Inhibitors 3. A Diastereomeric Approach to Chiral Nonracemic Tricyclic Ring Systems and the Discovery of Dolutegravir (S/GSK1349572) and (S/GSK1265744)

, 2013
Brian A. Johns, Takashi Kawasuji, Jason G. Weatherhead, Teruhiko Taishi, David P. Temelkoff, Hiroshi Yoshida, Toshiyuki Akiyama, Yoshiyuki Taoda, Hitoshi Murai, Ryuichi Kiyama, Masahiro Fuji, Norihiko Tánimoto, Jerry Jeffrey, Scott A. Foster, Tomokazu Yoshinaga, Takahiro Seki, Masanori Kobayashi, Akihiko Sato, Matthew N. Johnson, Edward P. Garvey, Tamio Fujiwara   +20 more
openalex   +1 more source

Therapeutic Opportunities in Infectious Diseases: Highlights from the Society of Medicines Research Symposium, held on March 14th 2013 at the National Heart & Lung Institute, London, UK [PDF]

, 2013
Alderton, W K, Anderson, Rosaleen, Collingwood, S P, Pryde, D C   +3 more
core   +1 more source

Structure-Guided Antiviral Peptides Identification Targeting the HIV-1 Integrase. [PDF]

ACS Phys Chem Au
Hossain MS, Alom MS, Kader MS, Hossain MA, Halim MA.   +4 more
europepmc   +1 more source

Emergence of Compensatory Mutations Reveals the Importance of Electrostatic Interactions between HIV-1 Integrase and Genomic RNA. [PDF]

mBio, 2022
Shema Mugisha C, Dinh T, Kumar A, Tenneti K, Eschbach JE, Davis K, Gifford R, Kvaratskhelia M, Kutluay SB.   +8 more
europepmc   +1 more source

Investigation on the sucrose binding pocket of HIV-1 Integrase by molecular dynamics and synergy experiments

, 2015
Cristina Tintori, Francesca Esposito, Francesca Morreale, Riccardo Martini, Enzo Tramontano, Maurizio Botta   +5 more
openalex   +1 more source

Systematic determination of in vitro phenotypic resistance to HIV-1 integrase strand transfer inhibitors from clinical samples [PDF]

, 2019
Aniqa Shahid, Wendy W. Zhang, Vincent Montoya, Peter K. Cheung, Natália Oliveira, Manraj S. Sidhu, Conan K. Woods, Marjorie Robbins, Chanson J. Brumme, P. Richard Harrigan   +9 more
openalex   +1 more source

HIV-1 integrase resistance associated mutations and the use of dolutegravir in Sub-Saharan Africa: A systematic review and meta-analysis. [PDF]

PLOS Glob Public Health, 2022
Ngoufack Jagni Semengue E, Santoro MM, Ndze VN, Ka'e AC, Yagai B, Nka AD, Dambaya B, Takou D, Teto G, Fabeni L, Colizzi V, Perno CF, Ceccherini-Silberstein F, Fokam J.   +13 more
europepmc   +1 more source

Quinolinonyl Derivatives as Dual Inhibitors of the HIV-1 Integrase Catalytic Site and Integrase-RNA interactions. [PDF]

ACS Med Chem Lett
Patacchini E, Madia VN, Albano A, Ruggieri G, Messore A, Ialongo D, Saccoliti F, Scipione L, Cosconati S, Koneru PC, Haney R, Kvaratskhelia M, Di Santo R, Costi R.   +13 more
europepmc   +1 more source

Synthesis of C3,C6-Diaryl 7-Azaindoles via One-Pot Suzuki-Miyaura Cross-Coupling Reaction and Evaluation of Their HIV-1 Integrase Inhibitory Activity. [PDF]

ACS Omega, 2023
Cardoza S, Yadav P, Ajmani A, Das P, Tandon V.   +4 more
europepmc   +1 more source

Crystal and Electronic Structures of Magnesium(II), Copper(II), and Mixed Magnesium(II)−Copper(II) Complexes of the Quinoline Half of Styrylquinoline-Type HIV-1 Integrase Inhibitors

, 2007
Blandine Courcot, D. Firley, Bernard Fraisse, P. Becker, Jean‐Michel Gillet, P. Pattison, Dmitry Chernyshov, Mehrez Sghaier, Fatima Zouhiri, Didier Desmaële, J. d'Angelo, F. Bonhomme, S. Geiger, Nour‐Eddine Ghermani   +13 more
openalex   +2 more sources