Results 161 to 170 of about 30,382,849 (226)

A computational overview of integrase strand transfer inhibitors (INSTIs) against emerging and evolving drug-resistant HIV-1 integrase mutants. [PDF]

Arch Microbiol, 2023
Sayyed SK, Quraishi M, Jobby R, Rameshkumar N, Kayalvizhi N, Krishnan M, Sonawane T.   +6 more
europepmc   +1 more source

Isolation of New Chemical Modulators of the Interaction Between HIV-1 Integrase and the Cellular Restriction Factor GCN2. [PDF]

Viruses
Torres C, Lagadec F, Basyuk E, Recordon-Pinson P, Métifiot M.   +4 more
europepmc   +1 more source

A point mutation in HIV-1 integrase redirects proviral integration into centromeric repeats. [PDF]

Nat Commun, 2022
Winans S, Yu HJ, de Los Santos K, Wang GZ, KewalRamani VN, Goff SP.   +5 more
europepmc   +1 more source

TAR RNA Mimicry of INI1 and Its Influence on Non-Integration Function of HIV-1 Integrase. [PDF]

Viruses
Kalpana GV, Ernst E, Haldar S.
europepmc   +1 more source

Synthetic Approaches to a Key Pyridone-carboxylic Acid Precursor Common to the HIV-1 Integrase Strand Transfer Inhibitors Dolutegravir, Bictegravir, and Cabotegravir. [PDF]

Org Process Res Dev, 2023
Mahajan PS, Burke TR.
europepmc   +1 more source

Structural Impact of Ex Vivo Resistance Mutations on HIV-1 Integrase Polymers Induced by Allosteric Inhibitors. [PDF]

J Mol Biol
Montermoso S, Eilers G, Allen A, Sharp R, Hwang Y, Bushman FD, Gupta K, Duyne GV.   +7 more
europepmc   +1 more source

Structure-Guided Antiviral Peptides Identification Targeting the HIV-1 Integrase. [PDF]

ACS Phys Chem Au
Hossain MS, Alom MS, Kader MS, Hossain MA, Halim MA.   +4 more
europepmc   +1 more source

Quinolinonyl Derivatives as Dual Inhibitors of the HIV-1 Integrase Catalytic Site and Integrase-RNA interactions. [PDF]

ACS Med Chem Lett
Patacchini E, Madia VN, Albano A, Ruggieri G, Messore A, Ialongo D, Saccoliti F, Scipione L, Cosconati S, Koneru PC, Haney R, Kvaratskhelia M, Di Santo R, Costi R.   +13 more
europepmc   +1 more source

Lack of activity of HIV-1 integrase strand-transfer inhibitors on recombinase activating gene (RAG) activity at clinically relevant concentrations. [PDF]

Microbiol Spectr
Demirdjian S, Duong VN, Byrum JN, Nayak A, McKinney CB, Perry JK, Callebaut C, Rodgers KK, Falkard B, Feng JY.   +9 more
europepmc   +1 more source

Comprehensive Analysis of HIV-1 Integrase Resistance-Related Mutations in African Countries. [PDF]

Pathogens
Branda F, Giovanetti M, Sernicola L, Farcomeni S, Ciccozzi M, Borsetti A.   +5 more
europepmc   +1 more source