Results 141 to 150 of about 42,534 (266)

Biological and Structural Analyses of New Potent Allosteric Inhibitors of HIV-1 Integrase. [PDF]

Antimicrob Agents Chemother, 2023
Bonnard D, Le Rouzic E, Singer MR, Yu Z, Le Strat F, Batisse C, Batisse J, Amadori C, Chasset S, Pye VE, Emiliani S, Ledoussal B, Ruff M, Moreau F, Cherepanov P, Benarous R.   +15 more
europepmc   +1 more source

Prevalence of Primary Drug Resistance Against HIV-1 Integrase Inhibitors in Canada

, 2018
Hezhao Ji, Aileen P. Patterson, Tracy Taylor, Claudia Rank, Jessica Halverson, Rupert Capiña, James Brooks, Paul Sandstrom   +7 more
openalex   +1 more source

HIV-1 Integrase Strand Transfer Inhibitors and Neurodevelopment. [PDF]

Pharmaceuticals (Basel), 2022
Foster EG, Gendelman HE, Bade AN.
europepmc   +1 more source

A Critical Role of the C-terminal Segment for Allosteric Inhibitor-induced Aberrant Multimerization of HIV-1 Integrase [PDF]

, 2014
Nikoloz Shkriabai, Venkatasubramanian Dharmarajan, Alison Slaughter, Jacques J. Kessl, Ross C. Larue, Lei Feng, James R. Fuchs, Patrick R. Griffin, Mamuka Kvaratskhelia   +8 more
openalex   +1 more source

Mechanisms of HIV-1 integrase resistance to dolutegravir and potent inhibition of drug-resistant variants. [PDF]

Sci Adv, 2023
Li M, Oliveira Passos D, Shan Z, Smith SJ, Sun Q, Biswas A, Choudhuri I, Strutzenberg TS, Haldane A, Deng N, Li Z, Zhao XZ, Briganti L, Kvaratskhelia M, Burke TR, Levy RM, Hughes SH, Craigie R, Lyumkis D.   +18 more
europepmc   +1 more source

Symmetrical 1-pyrrolidineacetamide showing anti-HIV activity through a new binding site on HIV-1 integrase¹ [PDF]

, 2008
Li Du, Yaxue Zhao, Liu‐Meng Yang, Yong‐Tang Zheng, Yun Tang, Xu Shen, Hualiang Jiang   +6 more
openalex   +1 more source

Predicted antiviral activity of tenofovir versus abacavir in combination with a cytosine analogue and the integrase inhibitor dolutegravir in HIV-1-infected South African patients initiating or failing first-line ART [PDF]

, 2018
Anne Derache, Collins Iwuji, Siva Danaviah, Jennifer Giandhari, Anne‐Geneviève Marcelin, Vincent Cálvez, Túlio de Oliveira, François Dabis, Deenan Pillay, Ravindra K. Gupta   +9 more
openalex   +1 more source

Conformational aspects of HIV‐1 integrase inhibition by a peptide derived from the enzyme central domain and by antibodies raised against this peptide [PDF]

, 1999
Richard G. Maroun, Daniel Krebs, Mahmoud Roshani, Horea Porumb, Christian Auclair, Frédéric Troalen, Serge Fermandjian   +6 more
openalex   +1 more source

Investigating the role of matrix and integrase in the nuclear import of the HIV-1 genome

, 2021
Anna C. Hearps
openalex   +1 more source

Recent Developments in the Synthesis of HIV-1 Integrase Strand Transfer Inhibitors Incorporating Pyridine Moiety. [PDF]

Int J Mol Sci, 2023
Starosotnikov AM, Bastrakov MA.
europepmc   +1 more source