Results 151 to 160 of about 30,099 (284)

Repositioning HIV-1 Integrase Inhibitors for Cancer Therapeutics: 1,6-Naphthyridine-7-carboxamide as a Promising Scaffold with Drug-like Properties

, 2012
Li‐Fan Zeng, Yong Wang, Roza Kazemi, Shili Xu, Zhong-Liang Xu, Tino W. Sanchez, Liu-Meng Yang, Bikash Debnath, Srinivas Odde, Hua Xie, Yong‐Tang Zheng, Jian Ding, Nouri Neamati, Ya-Qiu Long   +13 more
openalex   +1 more source

Update on Adverse Effects of HIV Integrase Inhibitors. [PDF]

Curr Treat Options Infect Dis, 2019
Kolakowska A, Maresca AF, Collins IJ, Cailhol J.   +3 more
europepmc   +1 more source

Prevalence of Primary Drug Resistance Against HIV-1 Integrase Inhibitors in Canada

, 2018
Hezhao Ji, Aileen P. Patterson, Tracy Taylor, Claudia Rank, Jessica Halverson, Rupert Capiña, James Brooks, Paul Sandstrom   +7 more
openalex   +1 more source

A Critical Role of the C-terminal Segment for Allosteric Inhibitor-induced Aberrant Multimerization of HIV-1 Integrase [PDF]

, 2014
Nikoloz Shkriabai, Venkatasubramanian Dharmarajan, Alison Slaughter, Jacques J. Kessl, Ross C. Larue, Lei Feng, James R. Fuchs, Patrick R. Griffin, Mamuka Kvaratskhelia   +8 more
openalex   +1 more source

Therapeutic Opportunities in Infectious Diseases: Highlights from the Society of Medicines Research Symposium, held on March 14th 2013 at the National Heart & Lung Institute, London, UK [PDF]

, 2013
Alderton, W K, Anderson, Rosaleen, Collingwood, S P, Pryde, D C   +3 more
core   +1 more source

Pharmacokinetics of HIV-Integrase Inhibitors During Pregnancy: Mechanisms, Clinical Implications and Knowledge Gaps. [PDF]

Clin Pharmacokinet, 2019
van der Galiën R, Ter Heine R, Greupink R, Schalkwijk SJ, van Herwaarden AE, Colbers A, Burger DM.   +6 more
europepmc   +1 more source

Resistance to HIV Integrase Inhibitors: About R263K and E157Q Mutations. [PDF]

Viruses, 2018
Charpentier C, Descamps D.
europepmc   +1 more source

Predicted antiviral activity of tenofovir versus abacavir in combination with a cytosine analogue and the integrase inhibitor dolutegravir in HIV-1-infected South African patients initiating or failing first-line ART [PDF]

, 2018
Anne Derache, Collins Iwuji, Siva Danaviah, Jennifer Giandhari, Anne‐Geneviève Marcelin, Vincent Cálvez, Túlio de Oliveira, François Dabis, Deenan Pillay, Ravindra K. Gupta   +9 more
openalex   +1 more source

X-ray and molecular modelling in fragment-based design of three small quinoline scaffolds for HIV integrase inhibitors

, 2011
K. Majerz-Maniecka, Robert Musioł, Agnieszka Skórska-Stania, D. Tabak, Paweł K. Mazur, Barbara J. Oleksyn, Jarosław Polański   +6 more
openalex   +2 more sources

Design and synthesis of photoactivatable aryl diketo acid-containing HIV-1 integrase inhibitors as potential affinity probes

, 2004
Xuechun Zhang, Christophe Marchand, Yves Pommier, Terrence R. Burke   +3 more
openalex   +1 more source