Results 161 to 170 of about 30,099 (284)

Limited marginal utility of deep sequencing for HIV drug resistance testing in the age of integrase inhibitors [PDF]

, 2018
Ronit R. Dalmat, Negar Makhsous, Gregory Pepper, Amalia Magaret, Keith R. Jerome, Anna Wald, Alexander L. Greninger   +6 more
openalex   +1 more source

Docking, Synthesis and Biological Evaluation of NovelDiketoquinoline Analogues as HIV-1 Integrase Inhibitor

, 2019
Kishore D. Deo, I.J. Singhvi, Sachin Patil, Avinash V. Patil   +3 more
openalex   +1 more source

Chemical scaffold recycling: Structure-guided conversion of an HIV integrase inhibitor into a potent influenza virus RNA-dependent RNA polymerase inhibitor designed to minimize resistance potential

, 2022
P.J. Slavish, M.G. Cuypers, Mary Ashley Rimmer, Alireza Abdolvahabi, Trushar Jeevan, Gyanendra Kumar, Jamie Jarusiewicz, Sivaraja Vaithiyalingam, Jeremy C. Jones, John J. Bowling, Jeanine E. Price, Rebecca M. DuBois, Jaeki Min, Richard J. Webby, Zoran Ranković, Stephen W. White   +15 more
openalex   +1 more source

The A128T Resistance Mutation Reveals Aberrant Protein Multimerization as the Primary Mechanism of Action of Allosteric HIV-1 Integrase Inhibitors [PDF]

, 2013
Lei Feng, Amit Sharma, Alison Slaughter, Nivedita Jena, Yasuhiro Koh, Nikolozi Shkriabai, Ross C. Larue, Pratiq A. Patel, Hiroaki Mitsuya, Jacques J. Kessl, Alan Engelman, James R. Fuchs, Mamuka Kvaratskhelia   +12 more
openalex   +1 more source

Chemistry and Structure−Activity Relationship of HIV-1 Integrase Inhibitor Integracide B and Related Natural Products

, 2003
Sheo B. Singh, John G. Ondeyka, William A. Schleif, Peter J. Felock, Daria J. Hazuda   +4 more
openalex   +1 more source

Development and Validation of a Machine Learning Model for Identifying Novel HIV Integrase Inhibitors. [PDF]

Cureus
Mukuhlani BT.
europepmc   +1 more source

Single‐dose pharmacokinetics and safety of ACC017, a novel HIV integrase inhibitor, in healthy adult participants: A first‐in‐human study [PDF]

Chaoying Hu, Y. Li, Yijun Zhou, Dong Zhao, Hui‐Yu Sun, Bin Li, Jing Ji, F. Zhang, Hong Qin, X. Yun   +9 more
openalex   +1 more source

Author Correction: Analyses of HIV-1 integrase sequences prior to South African national HIV-treatment program and availability of integrase inhibitors in Cape Town, South Africa [PDF]

, 2018
Dominik Brado, Adetayo Emmanuel Obasa, George Mondinde Ikomey, Ruben Cloete, Kamalendra Singh, Susan Engelbrecht, Ujjwal Neogi, Graeme Brendon Jacobs   +7 more
openalex   +1 more source

Shorter Time to Discontinuation Due to Treatment Failure in People Living with HIV Switched to Dolutegravir Plus Either Rilpivirine or Lamivudine Compared with Integrase Inhibitor-Based Triple Therapy in a Large Spanish Cohort

, 2022
Ramón Teira, Helena Díaz-Cuervo, Filipa Aragão, Manuel Castaño, Alberto Romero-Palacios, Bernardino Roca, Marta Montero, Marı́a José Galindo, Maria Jose Muñoz-Sánchez, Núria Espinosa, Joaquim Peraire, Elisa Martínez, Belén de la Fuente, Peré Domingo, Elisabeth Deig, María Dolores Merino, Paloma Geijo, Vicente Estrada, María Antonia Sepúlveda, Josefina García, Juan Berenguer, Adrián Curran   +21 more
openalex   +1 more source

Exploring the Potential of HIV Integrase Inhibitors as Therapeutic Agents Against HSV and HCMV: A Molecular Docking Study. [PDF]

J Exp Pharmacol
Rao AM, Sm F, Somashekara D, Gayam PKR, Rahangdale RR, Patil SS, Hariharapura RC.   +6 more
europepmc   +1 more source