Results 131 to 140 of about 10,572 (203)

Anticonvulsant action of indazole

Anticonvulsant action of indazole
Here we report that indazole is characterized as a potential anticonvulsant, inhibiting pentylenetetrazole-, electroshock- and strychnine-induced convulsions in mice (ED50's: 39.9, 43.2 and 82.4mg/kg, respectively) but not bicuculline- and picrotoxin-induced convulsions.
openaire  

<i>N</i>-Heterocyclic Olefins of Pyrazole and Indazole. [PDF]

Org Lett
Zhu B, Woyciechowski R, Hübner EG, Lederle F, Schmidt A.   +4 more
europepmc   +1 more source

Study on Phase I Metabolic Processes and Metabolite Biomarker Identification of Synthetic Cannabinoids 5F-ADB-PINACA and 5F-ADBICA in Human Liver Microsomes and Zebrafish Model. [PDF]

Molecules
Li H, Zheng H, Zhong S, Zhao Y, Lin J, Su H, Qian Z, Wang Y.   +7 more
europepmc   +1 more source

Design, synthesis, and antiproliferative activity of new 5-ethylsulfonyl-indazole-3-carbohydrazides as dual EGFR/VEGFR-2 kinases inhibitors. [PDF]

J Enzyme Inhib Med Chem
Al-Wahaibi LH, Abou-Zied HA, Mahmoud MA, Youssif BGM, Bräse S, Rabea SM.   +5 more
europepmc   +1 more source

In vitro CB₁ receptor activity of halogenated indazole synthetic cannabinoid receptor agonists. [PDF]

Arch Toxicol
Green H, McKenzie C, Hamra E, Rautio T, Wu X, Juneskog E, Sandblom R, Monti MC, Persson M, Norman C.   +9 more
europepmc   +1 more source

Synthetic cannabinoid receptor agonists containing silicon: exploring the metabolic pathways of ADMB- and Cumyl-3TMS-PrINACA in human urine specimens and post mortem material compared to in vitro and in silico data. [PDF]

Arch Toxicol
Zschiesche A, Carlier J, Pietsch J, Scheu M, Seibt J, Busardò FP, Auwärter V, Huppertz LM.   +7 more
europepmc   +1 more source

Arabidopsis P4-ATPases ALA1 and ALA7 Enhance Resistance to <i>Verticillium dahliae</i> via Detoxifying Vd-Toxins. [PDF]

Biology (Basel)
Wang F, Qiu M, Yao X, Li J, Ren H, Su M, Shen J, Li C, Jiang Q, Zhang Z, Li Y, Tang J, Li X, Fan Y, Pei Y.   +14 more
europepmc   +1 more source

New indazolebisphosphonates for bone targeted radiotherapy: synthesis, radiolabeling, in vitro and in vivo studies [PDF]

, 2008
Antunes, Inês F., Bilewicz, A., Gano, L., Majkowska, A., Neves, M., Santos, A., Teixeira, Fatima   +6 more
core  

C-to-N atom swapping and skeletal editing in indoles and benzofurans. [PDF]

Nature
Wang Z, Xu P, Guo SM, Daniliuc CG, Studer A.   +4 more
europepmc   +1 more source

[Simultaneous determination of 38 indazole amides synthetic cannabinoids and 15 metabolites in wastewater by solid phase extraction-liquid chromatography-tandem mass spectrometry]. [PDF]

Se Pu
Yang Z, Jiang LW, Wu YD, Jia R, Lyu JX.
europepmc   +1 more source