Results 161 to 170 of about 10,572 (203)

Development of a Buchwald-Hartwig Amination for an Accelerated Library Synthesis of Cereblon Binders. [PDF]

ACS Med Chem Lett
Lejava A, Miseo GA, Phan T, Zhu J, Powers HL, Li J, Mortensen DS, Zapf CW, Khambatta G, Buenviaje J, Holmberg-Douglas N.   +10 more
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Identification of Indazole- and Azaindazole-Substituted Cyclopentapyrroles as G2019S Leucine-Rich Repeat Kinase 2 Inhibitors for the Treatment of CNS Disorders. [PDF]

ACS Med Chem Lett
Feng S, Liang SH.
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Zur Kenntnis der Indazole

, 1946
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Inhibition of NLRP3 by a CNS-penetrating indazole scaffold

Torp J, Ferber D, Buthmann H, Hagelueken G, Deshpande A, Hartman G, Hughes RE, Salazar T, Tronnes S, Duisembekova A, Marleaux M, Hochheiser IV, Coll RC, Montgomery R, Fortney K, Py BF, Wilhelmsen K, Geyer M.   +17 more
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C3-INDAZOLE FUNCTIONALIZATION: A REVIEW

Targets in Heterocyclic Systems, 2021
Syntheses of nitrogen heteroaromatic systems are developed for numerous potential applications, particularly as biologically active compounds. Thus, scaffolds such as pyridinones,1 pyridoquinazolines,2 or indazoles (Figure 1) are frequently observed in the structure of biologically active compounds such as protein kinases inhibitors.3 Therefore, their ...
Giraud, F., Anizon, F., Moreau, P.
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Anticonvulsant action of indazole

Epilepsy Research, 2013
Here we report that indazole is characterized as a potential anticonvulsant, inhibiting pentylenetetrazole-, electroshock- and strychnine-induced convulsions in mice (ED50's: 39.9, 43.2 and 82.4 mg/kg, respectively) but not bicuculline- and picrotoxin-induced convulsions.
Nobuko, Matsumura, Kazue, Kikuchi-Utsumi, Kentaro, Sakamaki, Masahiko, Watabe, Koji, Aoyama, Toshio, Nakaki   +5 more
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Enthalpy of formation for indazoles (indazole, 1H-indazole-3-carboxylic acid, 1H-indazole-5-carboxylic acid, 1H-indazole-6-carboxylic acid and 1-methyl-1H-indazole-6-carboxylic methyl ester): experimental and theoretical studies

Journal of Thermal Analysis and Calorimetry, 2019
The molar standard enthalpy of formation in condensed and gas phases of indazole, 1H-indazole-3-carboxylic acid, 1H-indazole-5-carboxylic acid, 1H-indazole-6-carboxylic acid and 1-methyl-1H-indazole-6-carboxylic methyl ester is reported. These properties were obtained indirectly from experimental determinations of the compounds using isoperibolic ...
E. Orozco-Guareño, J. Baudelio Campos, Maximiliano Bárcena-Soto, Bernardo Zúñiga-Gutierrez   +3 more
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Synthesis of fused bis-indazoles/indazoles via a one-pot sequential strategy

Organic & Biomolecular Chemistry, 2023
An unprecedented protocol has been developed for the synthesis of fused bis-indazoles/indazoles via a one-pot sequential strategy.
Kishan Gugulothu, Ramanna Jatoth, Peramalla Edukondalu, Anusha Vanga, Raghavender Matta, K. Shiva Kumar   +5 more
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