The access to a novel variety of 4-fluorinated isoxazoles bearing an aryl or alkyl group at the C-3 position and an acetal fragment at the C-5 position has been achieved through a direct fluorination using N-fluorobenzenesulfonimide (NFSI) with yields up
Bacheley, Lucas +3 more
doaj +1 more source
Synthesis of some isoxazoline, isoxazole and pyrazole carboxylic acids as the precursors of new 1,2-diacyl-1-alkylhydrazines [PDF]
A number of isoxazoline, isoxazole and pyrazole carboxylic acids or their esters has been synthesized via the 1,3-dipolar cycloaddition of corresponding nitrile oxides or diazomethane to unsaturated dipolarophiles.
Antonevich, I. P., Katok, Ya. M.
core
Synthesis and reactions of aminopropenes, which contains functional groups [PDF]
В рамках данной работы осуществлен синтез енаминов, содержащих остатки первичных, вторичных, третичных аминов, а также амидную и тиоамидную группы. Проведено комплексное исследование структуры полученных соединений с помощью спектральных методов, включая
Lugovik, K. I., Луговик, К. И.
core
Recent Advances in the Synthesis of 2-Substituted Oxetanes [PDF]
Bull, JA, Davis, O
core +1 more source
Synthesis of new 3,5-substiuted isoxazole derivatives possessing potential anti-aggregative activity
Two new compounds belonging to 3,5-substituted isoxazoles class were synthesized for the action mechanism investigation and the pharmacophore fragment determination of potential anti-aggregative compounds of this class.
O. V. Demina +8 more
doaj
One-pot and Regioselective Gold-Catalyzed Synthesis of 2-Imidazolyl-a-pyrazolylbenzenes from 1-Propargyl-1H-benzotriazoles, Alkynes and Nitriles hrough a-imino Gold(I) Carbene Complexes [PDF]
Ballesteros Gimeno, Alfredo +3 more
core +1 more source
Reaction of condensed cyclohexane isoxazolones with Grignard rea gents
Synthesis of new 2-acyl derivatives of 1,3-cyclohexanediones, various variants of their subsequent chemical transformation are relevant for organic and bioorganic chemistry, since it is known that a large number of such substances are bioactive.
Наталья G. Vasilyeva +2 more
doaj
Synthesis of isoxazoles and their hydrazinolysis to 5-aminopyrazoles: an approach to fluorescent derivatives. [PDF]
Ríos MC +3 more
europepmc +1 more source
Substituent Effects Govern the Efficiency of Isoxazole Photoisomerization to Carbonyl‑2<i>H</i>‑Azirines. [PDF]
Jackson KE +3 more
europepmc +1 more source
Sequential Formal (4 + 1)-Spirocycloaddition/Oxidative Cleavage between Indoles and <i>β</i>‑Nitrostyrenes: One-Pot Route to Benzamide-Containing (3),4,5-Substituted Isoxazoles. [PDF]
Arutiunov NA +5 more
europepmc +1 more source

