Results 131 to 140 of about 2,157,910 (222)

Effects of muscarinic receptor antagonists on cocaine discrimination in wild-type mice and in muscarinic receptor M₁, M₂, and M₄ receptor knockout mice

, 2017
Muscarinic M1/M4 receptor stimulation can reduce abuse-related effects of cocaine and may represent avenues for treating cocaine addiction. Muscarinic antagonists can mimic and enhance effects of cocaine, including discriminative stimulus (SD) effects ...
Thomsen, Morgane, Morgane Thomsen, Lauren Joseph, Joseph, Lauren   +3 more
core   +1 more source

HIGH GLUCOSE CONDITIONS INCREASE DETRUSOR CHOLINERGIC EXCITABILITY BY REDUCING CAVEOLAE-MEDIATED INHIBITION OF MUSCARINIC M2-RECEPTOR ACTIVATION IN THE URINARY BLADDER

Continence, 2023
V Cristofaro, J Carew, S Dasari, M Sullivan   +3 more
doaj   +1 more source

Role of M2 muscarinic receptor in epithelial ovarian carcinoma (EOC)

, 2018
Role of M2 muscarinic receptor in epithelial ovarian carcinoma (EOC) Marilena Taggi1, M. Falcinelli1, V. Cacciamani1, V. Di Paolo1, A. M. Tata2 R.
Tata A. M, Canipari R., Taggi M, Falcinelli M, Di Paolo V, Cacciamani V   +5 more
core  

Protean agonism at the muscarinic M2 receptor

, 2015
Protean agonism at the muscarinic M2 receptor De Min A. (1), Matera C. (2), Messerer R. (3), Dallanoce C. (2), Holzgrabe U. (3), Mohr K. (1) (1) University of Bonn Pharmacology and Toxicology - Bonn, Deutschland (2) University of Milan ...
A. De Min, K. Mohr, C. Matera, C.M.L. Dallanoce, R. Messerer, U. Holzgrabe   +5 more
core   +2 more sources

Synthesis and biological profile at muscarinic M2 and M3 receptor subtypes of some analogs of diphenidol

, 1996
The synthesis and the pharmacological evaluation at M2 and M3 muscarinic receptor subtypes of some analogs of diphenidol with a modified intermediate chain is reported. The butyl chain was rendered more rigid or more polar.
Recanatini M., Chiarini A., Varoli L., Burnelli S., Guarnieri A., Budriesi R.   +5 more
core   +1 more source

Allosteric interactions at the m1, m2 and m3 muscarinic receptor subtypes

, 1991
The purpose of our study was to investigate the interactions of allosteric antagonists at the individual m1, m2 and m3 muscarinic receptor subtypes. This was achieved through the use of transformed Chinese hamster ovary cells stably expressing the rat m1
Lee, N. H., El-Fakahany, E. E.
core  

Dualsteric Agonist for M2 Muscarinic Receptor Causes Oxidative Stress and Mitochondrial Alteration in Human Glioblastoma Cancer Stem Cells. [PDF]

J Neurochem
Guerriero C, De Nuccio C, Petrone M, Rinaldi T, Cirigliano A, Visentin S, Bernardo A, Conti L, Matera C, De Amici M, Dallanoce C, Tata AM.   +11 more
europepmc   +1 more source

Evidence for M2 Muscarinic Receptor Antagonist Delay of Myopia Development Through Activation of Kir3.4 Channel in the Retina of Guinea Pigs. [PDF]

Invest Ophthalmol Vis Sci
Zhou H, Zhou G, Yang Q, Niu J, Wang R, Liu H, Hou S, Bi H, Liao X.   +8 more
europepmc   +1 more source

Herbal Amara extract induces gastric fundus relaxation via inhibition of the M2 muscarinic receptor. [PDF]

Neurogastroenterol Motil
Piqué-Borràs MR, Röhrl J, Künstle G.
europepmc   +1 more source

Initial characterization of M₂-muscarinic receptor overexpressing mouse heart. [PDF]

Naunyn Schmiedebergs Arch Pharmacol
Gergs U, Buchwalow IB, Hofmann B, Myslivecek J, Janisova K, Hadova K, Schettler F, Keller M, Klimas J, Neumann J.   +9 more
europepmc   +1 more source