Preparation of penta-azole containing cyclopeptides: challenges in macrocyclization
Herein is described the synthesis of several analogs of the natural product IB-01211 from concatenated azoles, via a biomimetic pathway based on cyclization-oxidation of serine containing peptides combined with the Hantzsch synthesis.
Álvarez Domingo, Mercedes +5 more
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Genetically Encoded Lysine-Selective Photocyclization Enables Phage Display Selection of Cyclic Peptide Binders. [PDF]
Yang XQ +8 more
europepmc +1 more source
Enantiopure synthesis of uniform [<i>n</i>]cycloparaphenylene-pillar[5]arene multi-macrocycles and their chiroptical properties. [PDF]
Hansmann YS +4 more
europepmc +1 more source
Total Synthesis of Isoriccardin C and Isoriccardin D Based on a Hydroxyl-Directed Palladium-Catalyzed Intramolecular C-H Alkenylation. [PDF]
Losada P, Mascareñas JL, Gulías M.
europepmc +1 more source
Catechol-derived propargyl diol cyclizations with malonyl dichloride: substituent effects on the formation of macrocyclic esters and their hydrochlorinated adducts. [PDF]
Lefkaritis G +3 more
europepmc +1 more source
On-Resin Synthesis and Diversification of Macrocyclic Disulfide Bridge Peptidomimetics via Bifunctional 5-Iodo-1,4-Triazoles. [PDF]
Malone MA +4 more
europepmc +1 more source
Development of proteome-derived cyclic peptide libraries via ortho-phthalaldehyde-assisted cyclization. [PDF]
Wei Y +6 more
europepmc +1 more source
Total Synthesis of Marine Natural Product Sunshinamide via Macrolactonization. [PDF]
Lu Y +6 more
europepmc +1 more source
Transcriptome-guided discovery and active-site gatekeeper engineering of a Viola arcuata asparaginyl ligase with superior catalytic performance. [PDF]
Zou Q +9 more
europepmc +1 more source

