Results 151 to 160 of about 13,541 (253)
Muscarinic acetylcholine receptor M3 (CHRM3; HM3) [PDF]
Science-Business eXchange, 2012 openaire +1 more source
International Journal of Biomedical ScienceMuscarinic acetylcholine M receptors (mAChRs) belong to the G protein-coupled receptor (GPCR) superfamily and play a crucial role in regulating and controlling the release of acetylcholine (ACh). This review aims to focus on M3 receptor (M3R) subtype distribution, function, efficacy, and clinical applications.
Shi-wan-er Chen, Jie Wu
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Ligand-Induced Activation of the M3-Muscarinic Acetylcholine Receptor
This thesis explores the computer-aided drug design of the M3-muscarinic acetylcholine receptor in three chapters. The first chapter focuses on molecular docking to identify novel agonists using the ZINC12 library. A model of the M3 receptor was built based on the M2 receptor.
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Beneficial Metabolic Effects Caused by Persistent Activation of β-Cell M3 Muscarinic Acetylcholine Receptors in Transgenic Mice [PDF]
, 2010 Dinesh Gautam +10 more
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Chronic regulation of colonic epithelial secretory function by activation of G protein-coupled receptors. [PDF]
, 2011 BACKGROUND: Enteric neurotransmitters that act at G protein-coupled receptors (GPCRs) are well known to acutely promote epithelial Cl(-) and fluid secretion.
Bertelsen, Lone S +6 more
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Pronounced Conformational Changes following Agonist Activation of the M3 Muscarinic Acetylcholine Receptor [PDF]
, 2005 Sung‐Jun Han +7 more
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