Results 171 to 180 of about 55,054 (301)

Histamine via histamine H1 receptor enhances the muscarinic receptor-induced calcium response to acetylcholine in an enterochromaffin cell model. [PDF]

Clin Exp Pharmacol Physiol, 2022
Pfanzagl B, Pfragner R, Jensen-Jarolim E.   +2 more
europepmc   +1 more source

Muscarinic receptor activation stimulates B-50/GAP43 phosphorylation in isolated nerve growth cones [PDF]

, 1989
CO Van Hooff, PN De Graan, A.B. Oestreicher, WH Gispen   +3 more
openalex   +1 more source

Progress on the development of Class A GPCR‐biased ligands

British Journal of Pharmacology, Volume 182, Issue 14, Page 3249-3300, July 2025.
Class A G protein‐coupled receptors (GPCRs) continue to garner interest for their essential roles in cell signalling and their importance as drug targets. Although numerous drugs in the clinic target these receptors, over 60% GPCRs remain unexploited. Moreover, the adverse effects triggered by the available unbiased GPCR modulators, limit their use and
Paula Morales, Magdalena M. Scharf, Marcel Bermudez, Attila Egyed, Rafael Franco, Olivia K. Hansen, Nadine Jagerovic, Jan Jakubík, György M. Keserű, Dóra Judit Kiss, Pawel Kozielewicz, Olav Larsen, Maria Majellaro, Ana Mallo‐Abreu, Gemma Navarro, Rubén Prieto‐Díaz, Mette M. Rosenkilde, Eddy Sotelo, Holger Stark, Tobias Werner, Laura M. Wingler   +20 more
wiley   +1 more source

The Effect on Quality of Life of Therapeutic Plasmapheresis and Intravenous Immunoglobulins on a Population of Myalgic Encephalomyelitis/Chronic Fatigue Syndrome Patients with Elevated β-Adrenergic and M3-Muscarinic Receptor Antibodies-A Pilot Study. [PDF]

J Clin Med
Oesch-Régeni B, Germann N, Hafer G, Schmid D, Arn N.   +4 more
europepmc   +1 more source

Daidzein is the in vivo active compound of Puerariae Lobatae Radix water extract for muscarinic receptor-3 inhibition against overactive bladder. [PDF]

Front Pharmacol, 2022
Qiang Y, Bai L, Tian S, Ma Y, Xu P, Cheng M, Wu Y, Li X, Xue M, Zhou X.   +9 more
europepmc   +1 more source

Phosphorylation of the cardiac muscarinic receptor in intact chick heart and its regulation by a muscarinic agonist.

, 1986
Madan M. Kwatra, Marie Thérèse Hosey
openalex   +1 more source

Subtypes of muscarinic receptor on cholinergic nerves and atrial cells of chicken and guinea‐pig hearts [PDF]

, 1988
D. Jeck, R. Lindmar, Konrad Löffelholz, Michaela Wänke   +3 more
openalex   +1 more source

The path to the G protein‐coupled receptor structural landscape: Major milestones and future directions

British Journal of Pharmacology, Volume 182, Issue 14, Page 3225-3248, July 2025.
G protein‐coupled receptors (GPCRs) play a crucial role in cell function by transducing signals from the extracellular environment to the inside of the cell. They mediate the effects of various stimuli, including hormones, neurotransmitters, ions, photons, food tastants and odorants, and are renowned drug targets.
Małgorzata M. Kogut‐Günthel, Zeenat Zara, Alessandro Nicoli, Alexandra Steuer, Marta Lopez‐Balastegui, Jana Selent, Sanjai Karanth, Melanie Koehler, Antonella Ciancetta, Layara Akemi Abiko, Franz Hagn, Antonella Di Pizio   +11 more
wiley   +1 more source

Striatal Cholinergic Interneurons Control Physical Nicotine Withdrawal via Muscarinic Receptor Signaling. [PDF]

Adv Sci (Weinh)
Kim B, Kim HA, Woo J, Lee HJ, Kim TK, Min H, Lee CJ, Im HI.   +7 more
europepmc   +1 more source

RGS3L allows for an M₂ muscarinic receptor-mediated RhoA-dependent inotropy in cardiomyocytes. [PDF]

Basic Res Cardiol, 2022
Levay MK, Krobert KA, Vogt A, Ahmad A, Jungmann A, Neuber C, Pasch S, Hansen A, Müller OJ, Lutz S, Wieland T.   +10 more
europepmc   +1 more source