Results 201 to 210 of about 76,340 (268)

Discovery of BNC375, a Potent, Selective, and Orally Available Type I Positive Allosteric Modulator of α7 nAChRs

, 2019
Andrew J. Harvey, Thomas D. Avery, Laurent Schaeffer, Christophe Joseph, Belinda C. Huff, Rajinder Singh, Christophe Morice, Bruno Giethlen, Anton A. Grishin, Carolyn Coles, Peter Kolesik, Stéphanie Wagner, Emile Andriambeloson, B. Huyard, Etienne Poiraud, Dharam Paul, Susan O’Connor   +16 more
openalex   +2 more sources

Assessing species-specific neonicotinoid toxicity using cross-species chimeric nicotinic acetylcholine receptors in a Drosophila model. [PDF]

Sci Rep
Lassota A, Hodge JJL, Soller M.
europepmc   +1 more source

Understanding varenicline function via key receptor and ligand interactions.

Cell Rep Phys Sci
Aiken SG, Fiorito D, Harper M, Pikus G, Underhill J, Murray J, Rawlinson J, O'Donoghue AC, Gotti C, Lummis SCR, Minguez Viñas T, Viscarra F, Bermudez I, Gallagher T, Oliveira ASF.   +14 more
europepmc   +1 more source

Regulation of Melanogenesis in Skin Epidermal Keratinocytes via Activation of α7 Nicotinic Acetylcholine Receptor on the Expression of α-Melanocyte-Stimulating Hormone. [PDF]

FASEB J
Guo MS, Wang X, Xia Y, Wu J, Dilidaer A, Gao J, Dong TT, Tsim KWK.   +7 more
europepmc   +1 more source

Nicotinic Receptors in the Medial Habenula to Interpeduncular Nucleus Pathway: Modulators of Reward, Aversion and Emotion. [PDF]

Eur J Neurosci
Ciscato M, Chouvaeff M, Mourot A.
europepmc   +1 more source

Point-to-point ligand–receptor interactions across the subunit interface modulate the induction and stabilization of conformational states of alpha7 nAChR by benzylidene anabaseines

, 2013
Matthew Isaacson, Nicole A. Horenstein, Clare Stokes, William R. Kem, Roger L. Papke   +4 more
openalex   +2 more sources

Discriminative stimulus and hypothermic effects of some derivatives of the nAChR agonist epibatidine in mice

Psychopharmacology, 2014
Jesse S. Rodriguez, Colin S. Cunningham, F. Moura, P. Ondachi, F. Carroll, L. McMahon   +5 more
semanticscholar   +1 more source

The Biological and Prognostic Implications of the Nicotinic Acetylcholine Receptor α3, α5, and α7 Subunits in Oral Squamous Cell Carcinoma. [PDF]

Cancer Med
Lin CM, Lin LW, Chen TC, Ye YL, Chiang BL.   +4 more
europepmc   +1 more source

α-RgIA:  A Novel Conotoxin That Specifically and Potently Blocks the α9α10 nAChR^,

, 2006
Michael J. Ellison, Christian Haberlandt, María Eugenia Gómez‐Casati, Maren Watkins, Ana Belén Elgoyhen, J. Michael McIntosh, Baldomero M. Olivera   +6 more
openalex   +2 more sources

Activation of the α7 nicotinic acetylcholine receptor mitigates cognitive deficits in mice with sepsis-associated encephalopathy by inhibiting microglial pyroptosis. [PDF]

World J Emerg Med
Wang Q, Luo Q, Su Z, Xu Y, Peng L, Wen Y, Zeng H, Ding H.   +7 more
europepmc   +1 more source