Results 141 to 150 of about 32,424 (300)

Hydrogen atom transfer in the photochemical isomerization of hydrazones of 1,2,4-oxadiazole derivatives [PDF]

, 2021
Maurizio D’Auria
openalex   +1 more source

Synthesis and Antibacterial Evaluation of 5-Aminosalicylic Acid Derivatives

Applied Sciences
The anti-inflammatory scaffold 5-aminosalicylic acid, which is widely used in therapeutic applications, was chosen for the synthesis of N-[3-(hydrazinecarbonyl)-4-hydroxyphenyl]acetamide (1) to enhance its antibacterial properties.
Kazimieras Anusevičius, Jūratė Šiugždaitė, Birutė Sapijanskaitė-Banevič, Valentas Špiliauskas, Birutė Grybaitė, Livija Tubytė, Vytautas Mickevičius   +6 more
doaj   +1 more source

Bis-1,3,4-Oxadiazole Derivatives As Novel And Potential Urease Inhibitors; Synthesis, In Vitro, And In Silico Studies.

, 2022
Momin Khan
openalex   +1 more source

Design, Synthesis, and Biological Evaluation of Novel 5-Substituted-2-(3,4,5-trihydroxyphenyl)-1,3,4-oxadiazoles as Potent Antioxidants

, 2016
A novel series of 5-(5-substituted-1,3,4-oxadiazol-2-yl)benzene-1,2,3-triols (3n-z) was designed, synthesized, and evaluated for its potential antioxidant activities.
A. M. Rabie, Atif S. Tantawy, Sahar M. I. Badr   +2 more
semanticscholar   +1 more source

C-(2-Deoxy-D-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors [PDF]

, 2021
Bokor, Éva, Csupász, Tibor, Docsa, Tibor, Gergely, Pál, Somsák, László, Szennyes, Eszter, Tóth, Nóra   +6 more
core   +1 more source

INOVAÇÃO E PROPRIEDADE INTELECTUAL DOS 1,2,4-OXADIAZÓIS: UMA PROSPECÇÃO TECNOLÓGICA FUNDAMENTADA EM BASE DE DADOS DE PATENTES E PERIÓDICOS

Química Nova
1,2,4-Oxadiazoles are heterocyclic compounds that have a remarkable range of applications. This overview focused on investigating the potential and scientific and technological evolution of these compounds through an analysis of patent databases and ...
Erick Caique Santos Costa, Jucleiton José Rufino de Freitas, Juliano Carlo Rufino Freitas   +2 more
doaj   +1 more source

Synthesis of biologically active enones: 2,3-dihydro-1,3,4-oxadiazoles, α-X-cyclopentenones and attempts towards limnophilaspiroketone and zerumbone [PDF]

, 2016
Anas J. Rasras
openalex   +1 more source

Modular and Computational Access to Innocuous Multistep Metal-Free Synthesis of 1,3,4-Oxadiazoles as Enzyme Inhibitors

, 2023
Muhammad Umair, Azizur Rehman, Muhammad Athar Abbasi, Sabahat Zahra Siddiqui, Javed Iqbal, Hira Khalid, Shahid Rasool, Shafi Ullah Khan, Fatiqa Zafar   +8 more
openalex   +1 more source

Microwave Irradiation Promoted Reactions of Orthoesters with Carboxylic Acid Hydrazides. Preparation of 1,3,4-Oxadiazoles [PDF]

Iranian Journal of Chemistry & Chemical Engineering, 1997
Rapid and highly efficient synthesis of 2- or 2,5-substituted 1,3,4-oxadiazoles by the condensation of aryl carboxylic acid hydrazides and orthoesters can be achieved under microwave irradiation using an unmodified commercial over in unsealed vessels.
Mohammad Sadegh Khajavi, Seyed Saheb Sadat Hosseini, Fatemeh Sefidkon   +2 more
doaj  

Molecular Docking Studies of 2-Mercapto-5-(3-Methoxyphenyl) 1, 3, 4 Oxadiazole Thiones with Focal Adhesion Kinase [PDF]

, 2014
The main objective of the present work is to perform molecular docking studies of the ligand 2- Mercapto-5-(3-Methoxy phenyl) 1,3,4 oxadiazole with protein focal adhesion kinase. A good correlation was observed in binding affinity of this complex.
Guruprasad, R., Kiran, K.S., Kokila, M.K.   +2 more
core