Results 191 to 200 of about 195,829 (332)

5-HT_1A Partial Agonist Tandospirone for Behavioral and Psychological Symptoms in Oldest-old Patients with Dementia at a Special Elderly Nursing Home. [PDF]

Clin Psychopharmacol Neurosci, 2021
Ochi S, Mori T, Iga JI, Ueno SI.
europepmc   +1 more source

Deoxyribose analogues of N⁶‐cyclopentyladenosine (CPA): partial agonists at the adenosine A₁ receptor in vivo [PDF]

, 1995
Ron A. A. Mathôt, Eleonora M. van der Wenden, W. Soudijn, Adriaan P. IJzerman, Meindert Danhof   +4 more
openalex   +1 more source

Metal‐Ligand Complexes as Multifunctional Platforms for Photo‐Activated Cancer Therapy

Advanced Science, EarlyView.
Metal‐ligand complexes serve as multifunctional platforms for photo‐activated cancer therapy, facilitating photothermal and photodynamic effects through light absorption and reactive oxygen species generation. This review categorizes these complexes by ligand and metal types, examines their roles in combined therapeutic approaches, and explores ...
Jeonga Kim, Saehan Choi, Yoonsung Nam
wiley   +1 more source

Partial Agonist Activity of Neonicotinoids on Rat Nicotinic Receptors: Consequences over Epinephrine Secretion and In Vivo Blood Pressure. [PDF]

Int J Mol Sci, 2021
Park J, Taly A, Bourreau J, De Nardi F, Legendre C, Henrion D, Guérineau NC, Legros C, Mattei C, Tricoire-Leignel H.   +9 more
europepmc   +1 more source

The profile of sabcomeline (SB‐202026), a functionally selective M₁ receptor partial agonist, in the marmoset [PDF]

, 1998
Mark H Harries, Nolwenn Samson, Jackie Cilia, A. J. Hunter   +3 more
openalex   +1 more source

Covalent Organic Frameworks‐Delivered Reuterin Drives Trained Immunity in Tumor‐Associated Macrophages to Enhance Melanoma Immunotherapy via Glycerophospholipid Metabolism

Advanced Science, EarlyView.
Covalent organic framework (COF)‐reuterin induces trained immunity in tumor‐associated macrophages, promoting the generation of nitric oxide and reactive oxygen species, thereby enhancing the antitumor immune response. Additionally, COF‐Reuterin directly kills tumor cells while simultaneously eradicating pathogenic intratumoural bacteria.
Jian‐Gang Zhang, Xiao‐Mei Zhang, Xi Wu, Cheng‐Kai Zhou, Zhen‐Zhen Liu, Xue‐Yue Luo, Liang Zhang, Wei Chen, Yong‐Jun Yang   +8 more
wiley   +1 more source

Regulation of calcium transients and isometric contractions by beta-1 adrenoceptor partial agonist denopamine in aequorin-injected dog right ventricular trabeculae

, 1992
Minoru Kohi, Masao Endoh
openalex   +1 more source

(+)‐WAY 100135, a partial agonist, at native and recombinant 5‐HT_1B/1D receptors [PDF]

, 1997
Colin Davidson, Michael Ho, Gary Price, Brian Jones, Jonathan A. Stamford   +4 more
openalex   +1 more source

KRAS mRNA Spleen‐Targeting Lipid Nanoparticles Synergize with Irinotecan Silicasomes to Robustly Augment the Cancer Immunity Cycle in Pancreatic Cancer

Advanced Science, EarlyView.
To overcome pancreatic cancer's immunosuppressive barriers, this study explores a dual approach: triggering immunogenic tumor cell death at the primary tumor site with irinotecan‐loaded silicasomes and enhancing immune activation in the spleen using LNPs encapsulating tumor antigen mRNA and a TLR7/8 agonist.
Lijia Luo, Xiang Wang, Yu‐Pei Liao, Andre E. Nel   +3 more
wiley   +1 more source

Discovery of a Bradykinin B2 Partial Agonist Profile of Raloxifene in a Drug Repurposing Campaign. [PDF]

Int J Mol Sci, 2020
Gomez-Gutierrez P, Perez JJ.
europepmc   +1 more source