Assessing the effect of breed, age, and sex on muscarinic receptor distribution in atria and ventricles of turkeys. [PDF]
Schoeller C, Abraham G.
europepmc +1 more source
Walnut Peptide KG-7 Alleviates Scopolamine-Induced Memory Deficits and Enhances Paracellular Transport via Tight Junction Modulation in a Mouse Model. [PDF]
Li M +6 more
europepmc +1 more source
Striatal M<sub>4</sub> muscarinic receptors determine the biological rhythm of activity, with a supportive role of M<sub>1</sub> muscarinic receptors. [PDF]
Janisova K +3 more
europepmc +1 more source
Cholinergic Activation of Corticofugal Circuits in the Adult Mouse Prefrontal Cortex. [PDF]
Gulledge AT.
europepmc +1 more source
[Treatment of duodenal ulcer with pirenzepin].
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PLASMA AND BILIARY DISPOSITION OF PIRENZEPINE IN MAN
SUMMARY1. The binding of pirenzepine, a selective muscarinic receptor antagonist to plasma and bile, was studied in vitro and in vivo. Plasma and hepatic bile were incubated with 14C‐pirenzepine and the bound fraction of 14C‐pirenzepine determined by equilibrium dialysis. The bound fractions were 12.6% (s.e.m.
Lee, SP, Paxton, JW, Choong, YS
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Pirenzepine in Erosive Duodenitis
Scandinavian Journal of Gastroenterology, 1985M Guslandi, A Tittobello
exaly +2 more sources
Pyrimidobenzodiazepines. Synthesis of pirenzepine analog.
Die Pharmazie, 1990The synthesis of Pyrimido[4,5-b][1,5]benzodiazepine derivatives from 4-(o-aminophenylene)amino-5-ethoxy-carbonyl-1,2-dihydro-6-methyl-2 - oxopyrimidine has been described. Pyrimidobenzodiazepine 5 alkylated with N-methyl-N'-chloroacetyl-piperazine gives a product related to pirenzepine. Compound 5 shows weak antianxiety and antidepressive action.
Długosz, Anna, Machoń, Zdzisław
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Pirenzepine and Gastrointestinal Motility: Differential Effect of Pirenzepine in the Gut
1985The capacity of pirenzepine to reduce gastric acid secretion in the basal state and after various forms of stimulation is well established by now (Jaup 1981). It is still under discussion whether the ulcer-healing and symptom-relieving effect of pirenzepine is solely due to the moderate acid reduction observed or whether other pharmacological ...
R. W. Stockbrügger +3 more
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Central oxotremorine antagonist properties of pirenzepine
Life Sciences, 1988Pirenzepine, the prototype M1 muscarinic receptor antagonist, is an important compound for investigating the functional significance of M1 receptors at the integrated level of behavior but may have limitations imposed by its physical chemistry. Like the nonselective antagonist methylatropine, pirenzepine is highly hydrophilic and crosses the blood ...
J M, Witkin +3 more
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